Inhibition of High‐Affinity Choline Uptake and Acetylcholine Synthesis by Quinuclidinyl and Hemicholinium Derivatives

Journal of Neurochemistry

Volumn 46, Issue 4, 1986, Pages 1170-1175

  Sterling, Gerald H ^a   Doukas, Peter H ^b,c   Ricciardi, Fiori J ^c   Biedrzycka, Diane W ^a   O'Neill, John J ^b  

^a DREXEL UNIVERSITY COLLEGE OF MEDICINE   (United States)

^b TEMPLE UNIVERSITY SCHOOL OF MEDICINE   (United States)

^c TEMPLE UNIVERSITY SCHOOL OF PHARMACY   (United States)

Author keywords

Acetylcholine; Choline uptake; Hemicholiniums; Quinuclidines

Indexed keywords

3 QUINUCLIDINOL; ACETYLCHOLINE; ACETYLCHOLINE IODIDE H 3; CHOLINE; CHOLINE H 3; DIPICRYLAMINE; GLUCOSE C 14; HEMICHOLINIUM 3; HEMICHOLINIUM DERIVATIVE; QUINUCLIDINE DERIVATIVE; RADIOISOTOPE; TROMETAMOL; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BRAIN; CENTRAL NERVOUS SYSTEM; DRUG ACCUMULATION; DRUG TISSUE LEVEL; NERVOUS SYSTEM; NONHUMAN; PRIORITY JOURNAL; RAT; STRUCTURE ACTIVITY RELATION; SYNAPTOSOME;

ACETYLCHOLINE; ANIMALS; BIOLOGICAL TRANSPORT; BRAIN; CEREBRAL CORTEX; CHOLINE; HEMICHOLINIUM 3; KINETICS; MALE; QUINUCLIDINES; RATS; RATS, INBRED STRAINS; SODIUM; STRUCTURE-ACTIVITY RELATIONSHIP; SYNAPTOSOMES; TEMPERATURE;

ANIMALIA;

EID: 0022469937     PISSN: 00223042     EISSN: 14714159     Source Type: Journal    
DOI: 10.1111/j.1471-4159.1986.tb00633.x     Document Type: Article

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