Intrinsic activity and effects of guanyl-5′-yl imidodiphosphate, Gpp(NH)p and sodium ion on the affinity of dynorphin 1-13, nalorphine and nalorphine-7,8-oxide to kappa-opioid receptor

General Pharmacology

Volumn 16, Issue 6, 1985, Pages 617-619

  Takayanagi, I ^a   Okumura, K ^a   Konno, F ^a   Koike, K ^a   Cho, N ^a,b   Hirobe, M ^a,b  

^a TOHO UNIVERSITY   (Japan)

^b UNIVERSITY OF TOKYO   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

DYNORPHIN; DYNORPHIN[1-13]; ETHYLKETAZOCINE H 3; GUANYLYLIMIDODIPHOSPHATE; NALORPHINE; NALORPHINE 7,8 OXIDE; NALOXONE; OPIATE; OPIATE RECEPTOR; RADIOISOTOPE; SODIUM; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BRAIN; CENTRAL NERVOUS SYSTEM; CYTOLOGY; DRUG ADMINISTRATION; DRUG MONITORING; DRUG RECEPTOR BINDING; GUINEA PIG; MALE GENITAL SYSTEM; MOUSE; NONHUMAN; PHARMACOKINETICS; PRELIMINARY COMMUNICATION; PRIORITY JOURNAL; VAS DEFERENS;

ANIMALS; BINDING, COMPETITIVE; BRAIN; CYCLAZOCINE; DYNORPHINS; ETHYLKETOCYCLAZOCINE; GUANOSINE TRIPHOSPHATE; GUANYLYL IMIDODIPHOSPHATE; MALE; MICE; MICE, INBRED STRAINS; MUSCLE CONTRACTION; MUSCLE, SMOOTH; NALORPHINE; NALOXONE; PEPTIDE FRAGMENTS; RATS; RECEPTORS, OPIOID; RECEPTORS, OPIOID, KAPPA; SODIUM; SYNAPTOSOMES; VAS DEFERENS;

EID: 0022397134     PISSN: 03063623     EISSN: None     Source Type: Journal    
DOI: 10.1016/0306-3623(85)90153-3     Document Type: Article

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