Alpha-adrenolytic properties of apogalanthamine and azapetine analogs

Journal of Pharmacobio-Dynamics

Volumn 8, Issue 11, 1985, Pages 917-923

  Watanabe, Kozo ^b   Sasaki, Yuji ^a   Kimura, Yukio ^a  

^a UNIVERSITY OF TOKUSHIMA   (Japan)

^b OTSUKA PHARMACEUTICAL CO LTD   (Japan)

Author keywords

6 methyl 5,6,7,8 tetrahydrodibenz c,e azocine; a2 adrenolytic; aj adrenolytic; apoglanthamine; azapetine; clonidine; gunea pig ileum; human platelet aggregation; rat anococcygeus muscle; rat vas deferens

Indexed keywords

ADRENALIN; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA ADRENERGIC RECEPTOR STIMULATING AGENT; AZAPETINE; CLONIDINE; COCAINE; GUANETHIDINE; NORADRENALIN; PHENTOLAMINE; PRAZOSIN; TETRODOTOXIN; YOHIMBINE;

ADVERSE DRUG REACTION; ANIMAL CELL; APOGALANTAMINE; APOGALANTAMINE DERIVATIVE; AZAPETINE DERIVATIVE; BLOOD AND HEMOPOIETIC SYSTEM; DRUG COMPARISON; DRUG EFFICACY; DRUG MONITORING; DRUG RECEPTOR BINDING; DRUG SENSITIVITY; GUINEA PIG; HUMAN; HUMAN CELL; ILEUM; LARGE INTESTINE; MALE GENITAL SYSTEM; MUSCLE; NONHUMAN; PHARMACOKINETICS; RAT; REGIONAL PERFUSION; SMALL INTESTINE; THROMBOCYTE; THROMBOCYTE AGGREGATION; VAS DEFERENS;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMAL; AZOCINES; CLONIDINE; DIBENZAZEPINES; DOSE-RESPONSE RELATIONSHIP, DRUG; EPINEPHRINE; GUINEA PIGS; HUMAN; ILEUM; IN VITRO; MALE; MUSCLE CONTRACTION; NOREPINEPHRINE; PLATELET AGGREGATION; RATS; RATS, INBRED STRAINS; VAS DEFERENS;

EID: 0022378882     PISSN: 0386846X     EISSN: None     Source Type: Journal    
DOI: 10.1248/bpb1978.8.917     Document Type: Article

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