Complete Conversion of Brain D2 Dopamine Receptors from the High‐ to the Low‐Affinity State for Dopamine Agonists, Using Sodium Ions and Guanine Nucleotide

Journal of Neurochemistry

Volumn 44, Issue 6, 1985, Pages 1925-1935

  Grigoriadis, Dimitri ^a   Seeman, Philip ^a  

^a UNIVERSITY OF TORONTO   (Canada)

Author keywords

Binding affinity; D2 dopamine receptors; Guanine nucleotide; Rat striatum; Serotonin; Sodium ions; 3H Spiperone

Indexed keywords

2 AMINO 6,7 DIHYDROXYTETRALIN; CHOLINE; DOPAMINE; DOPAMINE RECEPTOR; DOPAMINE RECEPTOR STIMULATING AGENT; GUANINE NUCLEOTIDE; GUANYLYLIMIDODIPHOSPHATE; KETANSERIN; LITHIUM CHLORIDE; NORADRENALIN; POTASSIUM CHLORIDE; RADIOISOTOPE; SEROTONIN; SODIUM; SODIUM CHLORIDE; SULPIRIDE; TRYPTAMINE;

ANIMAL CELL; BIOLOGICAL MODEL; BRAIN; CENTRAL NERVOUS SYSTEM; DOSE RESPONSE; DRUG ANTAGONISM; DRUG COMPARISON; DRUG INTERACTION; DRUG RECEPTOR BINDING; DRUG RESPONSE; IN VITRO STUDY; NONHUMAN; PHARMACOKINETICS; PRIORITY JOURNAL; PROPYLNORAPOMORPHINE H 3; RAT; SPIPERONE H 3;

ANIMAL; APOMORPHINE; BRAIN; GUANINE NUCLEOTIDES; IN VITRO; KETANSERIN; MALE; PIPERIDINES; RATS; RATS, INBRED STRAINS; RECEPTORS, DOPAMINE; SODIUM; SPIPERONE; SUPPORT, NON-U.S. GOV'T; TETRAHYDRONAPHTHALENES; TRITIUM;

EID: 0021870454     PISSN: 00223042     EISSN: 14714159     Source Type: Journal    
DOI: 10.1111/j.1471-4159.1985.tb07189.x     Document Type: Article

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