Selective Inhibition of Thrombin by (2R,4R)-4-Methyl-l-[N2-[(3-methyl-l,2,3,4-tetrahydro-8-quinolinyl)sulfonyl]-L-arginyl)]-2-piperidinecarboxylic Acid

Biochemistry

Volumn 23, Issue 1, 1984, Pages 85-90

  Kikumoto, Ryoji ^a   Tamao, Yoshikuni ^a   Tezuka, Toru ^a   Tonomura, Shinji ^a   Hara, Hiroto ^a   Ninomiya, Kunihiro ^a   Hijikata, Akiko ^b   Okamoto, Shosuke ^b  

^a MITSUBISHI CHEMICAL CORPORATION   (Japan)

^b KOBE UNIVERSITY SCHOOL OF MEDICINE   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ARGATROBAN; ARGININE DERIVATIVE; BLOOD CLOTTING FACTOR 10A; HEPARIN; KALLIKREIN; PLASMIN; THROMBIN; THROMBIN DERIVATIVE; TRYPSIN;

DRUG COMPARISON; DRUG INTERACTION; ENZYME INHIBITION; KALLIKREIN BLOOD LEVEL; NONHUMAN; STRUCTURE ACTIVITY RELATION; THEORETICAL STUDY;

ANIMALS; BINDING SITES; BINDING, COMPETITIVE; CATTLE; KINETICS; OPTICAL ROTATION; PIPECOLIC ACIDS; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; THROMBIN;

BOVINAE;

EID: 0021327417     PISSN: 00062960     EISSN: 15204995     Source Type: Journal    
DOI: 10.1021/bi00296a014     Document Type: Article

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