Synthesis and characterization of iodinated vasopressin antagonists which retain high affinity for the vasopressin receptor

Biochemical and Biophysical Research Communications

Volumn 121, Issue 3, 1984, Pages 878-883

  Moore, Michael L ^a   Huffman, William F ^a   Roberts, Gerald D ^a   Rottschaefer, Susan ^a   Sulat, Lynn ^a   Stefankiewicz, James S ^a   Stassen, Frans ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ARGIPRESSIN; ARGIPRESSIN[2 (3 IODOTYROSINE)]; ARGIPRESSIN[2 (3,5 DIIODOTYROSINE)]; LYPRESSIN; UNCLASSIFIED DRUG; VASOPRESSIN ANTAGONIST; VASOPRESSIN RECEPTOR; VASOPRESSIN[1,9 N PENTAMETHYLENE 2 (3 IODO DEXTRO TYROSINE)]; VASOPRESSIN[1,9 N PENTAMETHYLENE 2 (3,5 DIIODO DEXTRO TYROSINE)]; VASOPRESSIN[1,9 N PENTAMETHYLENE 2 DEXTRO TYROSINE 4 VALINE];

ANIMAL CELL; ARTICLE; DRUG ANALYSIS; DRUG COMPARISON; DRUG IDENTIFICATION; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG STABILITY; DRUG SYNTHESIS; FISH; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; KIDNEY; MASS SPECTROMETRY; NONHUMAN; PHARMACOKINETICS; PRELIMINARY COMMUNICATION;

ARGININE VASOPRESSIN; CHEMISTRY; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; IODINE; MASS SPECTROMETRY; RECEPTORS, CELL SURFACE; RECEPTORS, VASOPRESSIN;

ANIMALIA;

EID: 0021270329     PISSN: 0006291X     EISSN: 10902104     Source Type: Journal    
DOI: 10.1016/0006-291X(84)90759-9     Document Type: Article

References (7)

1. Evaluation of an iodination procedure for arg8-vasopressin
2. [1-(.beta.-mercapto-.beta.,.beta.-cyclopentamethylenepropionic acid),2-(O-methyl)tyrosine]arginine-vasopressin and [1-(.beta.-mercapto-.beta.,.beta.-cyclopentamethylenepropionic acid)]arginine-vasopressin, two highly potent antagonists of the vasopressor response to arginine-vasopressin