SCOPUS 정보 검색 플랫폼

Biochemical and Biophysical Research Communications

Volumn 122, Issue 2, 1984, Pages 791-797

Azapeptides: A new class of angiotensin-converting enzyme inhibitors

(6) Greenlee, W J a Thorsett, E D a Springer, J P a Patchett, A A a Ulm, E H a Vassil, T C a

a MERCK RESEARCH LABORATORIES (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AZAPEPTIDE; CAPTOPRIL; DIPEPTIDYL CARBOXYPEPTIDASE; DIPEPTIDYL CARBOXYPEPTIDASE INHIBITOR; ENALAPRIL DERIVATIVE; ENALAPRILAT; N (2 PHENETHYLALANYL)PROLINAMIDE; UNCLASSIFIED DRUG;

ARTICLE; DRUG COMPARISON; DRUG PROTEIN BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; STRUCTURE ACTIVITY RELATION; THEORETICAL STUDY;

ANGIOTENSIN-CONVERTING ENZYME INHIBITORS; AZA COMPOUNDS; INDICATORS AND REAGENTS; PEPTIDES; PROTEIN CONFORMATION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0021149796 PISSN: 0006291X EISSN: 10902104 Source Type: Journal
DOI: 10.1016/S0006-291X(84)80103-5 Document Type: Article

Times cited : (39)

References (23)

2
- 0019448541
- (1981) Br. J. Clin. Pharmacol. , vol.11 , pp. 461-467
- Brunner¹ Desponds² Biollaz³ Keller⁴ Ferber⁵ Gavras⁶ Brunner⁷ Schnelling⁸

3
- 0015893576
- (1973) Experientia , vol.29 , pp. 947-948
- Oehme¹ Katzwinkel² Vogt³ Niedrich⁴

4
- 0016895991
- Polypeptides. Part XIV. A comparative study of the stability towards enzymes of model tripeptides containing ?-aza-amino-acids, L-amino-acids, and D-amino-acids
- (1976) Journal of the Chemical Society, Perkin Transactions 1 , vol.1 , pp. 244-248
- Dutta¹ Giles²

5
- 0017623248
- (1977) J. Med. Chem. , vol.20 , pp. 1464-1468
- Dorn¹ Zimmerman² Yang³ Yurewicz⁴ Ashe⁵ Frankshun⁶ Jones⁷

6
- 0019909012
- (1982) Z. Naturforsch. , vol.37 b , pp. 1075-1081
- Folkers¹ Bowers² Lutz³ Friebel⁴ Kubiak⁵ Schircks⁶ Rampold⁷

7
- 84915496076
- Chemistry and Biology of Peptides
- J. Meinhofer, Boston, 1972, Ann Arbor Science, NY
- (1972) Proc. 3rd Peptide Symp. , pp. 541-554
- Parry¹ Russel² Szelke³

8
- 0018132888
- (1978) J. Med. Chem. , vol.21 , pp. 1018-1024
- Dutta¹ Furr² Giles³ Valcaccia⁴

9
- 0016417266
- Polypeptides. Part XIII. Preparation of ?-aza-amino-acid (carbazic acid) derivatives and intermediates for the preparation of ?-aza-peptides
- (1975) Journal of the Chemical Society, Perkin Transactions 1 , pp. 1712-1720
- Dutta¹ Morley²

10
- 0012463647
- (1975) Tetrahedron , vol.31 , pp. 2940-2943
- Gray¹ Parker²

11
- 84916111794
- Berger, J. G. and Weinstein, J. (1981), European Patent Application 0054862 (Schering Corp.)

12
- 84916111793
- Berger, J. G. and Weinstein, J. (1981), European Patent Application 0054862 (Schering Corp.)

13
- 0017102431
- (1976) Ann. Rev. Biochem. , vol.45 , pp. 73-94
- Soffer¹

14
- 0018933572
- (1980) Biochem. Biophys. Res. Commun. , vol.93 , pp. 1290-1296
- Becker¹ Caprioli²

15
- 84916111792
- Bull, H. G., Thornberry, N. A., and Cordes, E. H., 1983, Merck Sharp and Dohme International Medical Advisory Council, “MEDAC” Strasbourg, June 5-7, 1983, proceedings.

16
- 0000363447
- This dihedral angle was claculated using the data of:
- (1981) J. Mol. Struct. , vol.72 , pp. 217-231
- Fernholt¹ Samdal² Seip³

17
- 84912909482
- Peptides: Structure and Function
- V.J. Hruby, D.H. Rich, Pierce Chem. Co., Ann Arbor, MI
- (1983) proc. of 8th Am. Peptide Symp. , pp. 555-559
- Thorsett¹ Harris² Aster³ Peterson⁴ Tristram⁵ Snyder⁶ Springer⁷ Patchett⁸

18
- 84916111791
- 50 = 7.4 uM.

19
- 84916111790
- Recently bicyclic lactam inhibitors with ψ as large as 200° have been reported (12).

20
- 0012046737
- Peptides: Structure and Function
- V.J. Hruby, D.H. Rich, Pierce Chem. Co., Rockford, Il
- (1983) proc. of 8th Am. Peptide Symp. , pp. 551-554
- Wyvratt¹ Tischler² Ikeler³ Springer⁴ Tristram⁵ Patchett⁶

21
- 37049123264
- 13C nuclear magnetic resonance spectroscopy and cis/trans isomerism in dipeptides containing proline
- (1972) Journal of the Chemical Society, Chemical Communications , pp. 994
- Thomas¹ Williams²

22
- 0016391484
- (1974) J. Amer. Chem. Soc. , vol.96 , pp. 7312-7317
- Evans¹ Rabenstein²

23
- 0020321280
- (1982) Med. Res. Rev. , vol.2 , pp. 1-41
- Petrillo¹ Ondetti²

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.