Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Nature

Volumn 302, Issue 5911, 1983, Pages 832-837

  Arrang, Jean Michel ^a   Garbarg, Monique ^a   Schwartz, Jean Charles ^a  

^a CENTRE PAUL BROCA   (France)

Author keywords

[No Author keywords available]

Indexed keywords

BRAIN RECEPTOR; BURIMAMIDE; CHLORPHENIRAMINE; CIMETIDINE; CYCLIC AMP; CYCLIZINE; DIMAPRIT; HISTAMINE; HISTAMINE RECEPTOR; IMPROMIDINE; MEPYRAMINE; METIAMIDE; N METHYLHISTAMINE; N,N DIMETHYLHISTAMINE; NEW DRUG; RADIOISOTOPE; RANITIDINE; SKF 91486; TIOTIDINE; UNCLASSIFIED DRUG;

ANIMAL CELL; BRAIN CORTEX; BRAIN SLICE; CENTRAL NERVOUS SYSTEM; DRUG ANTAGONISM; DRUG EFFICACY; DRUG INTERACTION; HISTAMINE H 3; METHYLHISTAMINE; NONHUMAN; RAT; SKF 91486;

ANIMAL; CEREBRAL CORTEX; HISTAMINE; HISTAMINE ANTAGONISTS; HISTAMINE RELEASE; IN VITRO; KINETICS; POTASSIUM; RATS; RECEPTORS, HISTAMINE; RECEPTORS, HISTAMINE H3; STRUCTURE-ACTIVITY RELATIONSHIP; SUPPORT, NON-U.S. GOV'T;

EID: 0020587209     PISSN: 00280836     EISSN: None     Source Type: Journal    
DOI: 10.1038/302832a0     Document Type: Article

References (38)

1. Weinreich, D. in Biochemistry of Characterised Neurons (ed. Osborne, C. Ν. Ν.) 153-175 (Pergamon, Oxford, 1977).
2. Schwartz, J. C, Pollard, H. & Quach, T. T. J. Neurochem. 35, 26-33 (1980).
3. Garbarg, M., Barbin, G., Feger, J. & Schwartz, J. C. Science 186, 833-835 (1974).
4. Barbin, G., Garbarg, M., Schwartz, J. C. & Storm-Mathisen, J. J. Neurochem. 26, 259-263 (1976).
5. Haas, H. L. & Wolf, P. Pflügers Arch. ges. Physiol. 362, 38 (1976).
6. Ash, A. S. F. & Schild, H. O. Br. J. Pharmac. Chemother. 27, 427-439 (1966).
7. Black, J. W., Duncan, W. A. M., Durant, C. J., Ganellin, C. R. & Parsons, M. E. Nature 236, 385-390 (1972).
8. Quach, T. T., Duchemin, A. M., Rose, C. & Schwartz, J. C. Molec. Pharmac. 17, 301-308 (1980).
9. Palacios, J. M., Garbarg, M., Barbin, G. & Schwartz, J. C. Molec. Pharmac. 14, 971-982 (1978).
10. Hegstrand, L. R., Kanof, P. D. & Greengard, P. Nature 260, 163-165 (1976).
11. Langer, S. Z. Br. J. Pharmac. 60, 481-498 (1977).
12. Starke, K. A. Rev. Pharmac. Tax. 21, 7-30 (1981).
13. Baudry, M., Martres, M. P. & Schwartz, J. C. J. Neurochem. 21, 1301-1309 (1973).
14. Garbarg, M., Barbin, G., Bischoff, S., Pollard, H. & Schwartz, J. C. Brain Res. 106, 333-348 (1976).
15. Barbin, G., Hirsch, J.-C, Garbarg, M. & Schwartz, J. C. Brain Res. 92, 170-174 (1975).
16. Verdière, M., Rose, C. & Schwartz, J. C. Eur. J. Pharmac. 34, 157-168 (1975).
17. Tuomisto, L., Tuomisto, J. & Walaszek, E. J. Med. Biol. 53, 40–46 (1975).
18. Subramanian, N. & Mulder, A. H. Eur. J. Pharmac. 35, 203-206 (1976).
19. Biggs, M. J. & Johnson, E. S. Br. J. Pharmac. 70, 555-560 (1980).
20. Subramanian, N. Life Sci. 31, 557-562 (1982).
21. Taylor, K. M. & Snyder, S. H. J. Neurochem. 21, 1215-1223 (1973).
22. Schwartz, J. C, Lampart, C. & Rose, C. J. Neurochem. 19, 801-810 (1972).
23. Schwartz, J. C, Larapart, C. & Rose, C. J. Neurochem. 17, 1527-1534 (1970).
24. Durant, G. J. et al. Nature 276, 403-405 (1978).
25. Cheng, Y. C. & Prusoff, W. H. Biochem. Pharmac. 22, 3099-3108 (1973).
26. Ganellin, C. R. in Pharmacology of Histamine Receptors (eds Ganellin, C. R. & Parsons, M. E.) 10-102 (Wright PSG, Bristol, 1982).
27. Schwartz, J. C. et al. in Pharmacology of Histamine Receptors (eds Ganellin, C. R. & Parsons, M. E.) 351-391 (Wright PSG, Bristol, 1982).
28. Yellin, T. O., Buck, S. H., Gilman, D. J., Jones, D. F & Wardleworth, J. M. Life Sci. 25, 2001-2009 (1979).
29. Parsons, M. E., Blakemore, R. C, Durant, G. J., Ganellin, C. R. & Rasmussen, A. C. Ag Actions 5, 464 (1975).
30. Trung Tuong, M. D., Garbarg, M. & Schwartz, J. C. Nature 287, 548-551 (1980).
31. Black, J. W., Gerskowitch, V. P. & Leff, P. in Pharmacology of Histamine Receptors (eds Ganellin, C. R. & Parsons, M. E.) 1-9 (Wright PSG, Bristol, 1982).
32. Dismukes, K., Rogers, M. & Daly, J. W. J. Neurochem. 26, 785-790 (1976).
33. Wemer, J., Van Der Lugt, J.-C, De Langen, C. D. J. & Mulder, A. H. J. Pharmac. exp. Ther. 211, 445-451 (1979).
34. Dolphin, A., Adrien, J., Hamon, M. & Bockaert, J. Molec. Pharmac. 15, 1-15 (1979).
35. Mounsey, I., Brady, K. A., Carroll, J., Fisher, R. & Middlemiss, D. N. Biochem. Pharmac. 31, 49-53 (1982).
36. Quach, T. T., Rose, C, Duchemin, A. M. & Schwartz, J. C. Nature 298, 373-375 (1982).
37. Snyder, S. H., Baldessarini, R. J. & Axelrod, J. J. Pharmac. exp. Ther 153, 544-549 (1966).
38. Parker, R. B. & Waud, D. R. J. Pharmac. exp. Ther. 177, 1-12 (1971).