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Volumn 39, Issue 15, 1983, Pages 2445-2458

A comparison of the antibacterial and β-lactamase inhibiting properties of penam and (2,3)-β-methylenepenam derivatives. The discovery of a new β-lactamase inhibitor. Conformational requirements for penicillin antibacterial activity

(5) Keith, D D a Tengi, J a Rossman, P a Todaro, L a Weigele, M a

a HOFFMANN LA ROCHE INC (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2,3 METHYLENEPENAM DERIVATIVE; ANTIINFECTIVE AGENT; BETA LACTAMASE; DRUG ANALOG; MECILLINAM; NEW DRUG; PENAM DERIVATIVE; PENICILLIN BINDING PROTEIN; PENICILLIN G; SULBACTAM; UNCLASSIFIED DRUG;

DRUG COMPARISON; DRUG EFFICACY; DRUG PROTEIN BINDING; DRUG SCREENING; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENTEROBACTERIACEAE; ENZYME INHIBITION; IN VITRO STUDY; INFRARED SPECTROMETRY; MICROCOCCACEAE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; PKA; STRUCTURE ACTIVITY RELATION;

BACTERIA (MICROORGANISMS); ENTEROBACTERIACEAE; MICROCOCCACEAE;

EID: 0020518162 PISSN: 00404020 EISSN: None Source Type: Journal
DOI: 10.1016/S0040-4020(01)92137-4 Document Type: Article

Times cited : (35)

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