2-Benzodioxinylaminoethanols: A New Class of β-Adrenergic Blocking and Antihypertensive Agents

Journal of Medicinal Chemistry

Volumn 24, Issue 8, 1981, Pages 994-998

  Lalloz, Lucien ^a   Loppinet, Vincent ^a   Coudert, Gérard ^a   Guillaumet, Gérald ^a   Loubinoux, Bernard ^a   Labrid, Claude ^b   Beaughard, Michele ^b   Dureng, Georges ^b   Claude Lamar, Jean ^b  

^a UNIVERSITÉ DE LORRAINE   (France)

^b CERM Centre Europeen de Recherches Mauvernay   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ISOPRENALINE; PRACTOLOL; PROPRANOLOL;

(2 BENZODIOXANYL)ETHANOLAMINE DERIVATIVE; 1 (1,4 BENZODIOXIN 2 YL) 2 [4 (2 METHOXYPHENYL)PIPERAZINO]ETHANOL; 2 BENZODIOXINYLAMINOETHANOL DERIVATIVE; ANIMAL EXPERIMENT; BETA ADRENERGIC RECEPTOR BLOCKING; BLOOD PRESSURE; CARDIOVASCULAR SYSTEM; DOSE RESPONSE; DRUG ANALYSIS; DRUG ANTAGONISM; DRUG COMPARISON; DRUG RESPONSE; DRUG SCREENING; DRUG SYNTHESIS; GUINEA PIG; HEART; HEART ATRIUM; HYPERTENSION; IN VITRO STUDY; INFRARED SPECTROMETRY; INTRAVENOUS DRUG ADMINISTRATION; NUCLEAR MAGNETIC RESONANCE; RAT; RESPIRATORY SYSTEM; SPONTANEOUSLY HYPERTENSIVE RAT; THEORETICAL STUDY; TRACHEA;

ADRENERGIC BETA-ANTAGONISTS; ANIMAL; ANTIHYPERTENSIVE AGENTS; DIOXINS; DOSE-RESPONSE RELATIONSHIP, DRUG; GUINEA PIGS; HYPERTENSION; IN VITRO; MALE; MUSCLE CONTRACTION; MUSCLE, SMOOTH; MYOCARDIAL CONTRACTION; RATS; RATS, MUTANT STRAINS; TRACHEA;

EID: 0019831633     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00140a015     Document Type: Article

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