Inhibitory effect of amidino-substituted heterocyclic compounds on the amidase activity of plasmin and of high and low molecular weight urokinase and on urokinase-induced plasminogen activation

Thrombosis Research

Volumn 24, Issue 1-2, 1981, Pages 73-83

  Geratz, J D ^a   Shaver, S R ^a   Tidwell, R R ^a  

^a UNIVERSITY OF NORTH CAROLINA SCHOOL OF MEDICINE   (United States)

Author keywords

Amidines; plasmin inhibitors; urokinase inhibitors

Indexed keywords

4 AMINOBENZAMIDINE; AMIDASE; AMIDINE; BENZAMIDINE; DIAMIDINE DERIVATIVE; PLASMIN; PLASMINOGEN; PLASMINOGEN ACTIVATOR; PLASMINOGEN ACTIVATOR INHIBITOR; UROKINASE;

BLOOD AND HEMOPOIETIC SYSTEM; ENZYME INHIBITION; HUMAN CELL; IN VITRO STUDY;

AMIDINES; AMIDOHYDROLASES; BENZAMIDINES; ENDOPEPTIDASES; HETEROCYCLIC COMPOUNDS; HUMAN; HYDROGEN-ION CONCENTRATION; INDOLES; MOLECULAR WEIGHT; PLASMIN; PLASMINOGEN ACTIVATORS; SUPPORT, NON-U.S. GOV'T; SUPPORT, U.S. GOV'T, P.H.S.; URINARY PLASMINOGEN ACTIVATOR;

EID: 0019787830     PISSN: 00493848     EISSN: None     Source Type: Journal    
DOI: 10.1016/0049-3848(81)90033-5     Document Type: Article

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6. Amidino-substituted heterocycles as probes of the specificity pocket of trypsin-like proteases
7. The isolation and characterization of plasminogen activators (urokinase) from human urine
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