3-Substituted 5,7-Dimethylpyrazolo[1,5-α]pyrimidines, 3′,5′-Cyclic amp Phosphodiesterase Inhibitors

Journal of Medicinal Chemistry

Volumn 17, Issue 6, 1974, Pages 645-648

  Novinson, Thomas ^a   Hanson, Ruth ^a   Dimmitt, K ^a   Simon, Lionel N ^a   Robins, Roland K ^a   O'Brien, Darrell E ^a  

^a Valeant Pharmaceuticals International   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CYCLIC AMP; CYCLIC AMP PHOSPHODIESTERASE; PHOSPHODIESTERASE; PYRAZOLO[1,5 A]PYRIMIDINE DERIVATIVE; PYRAZOLOPYRIMIDINE DERIVATIVE;

CATTLE; DRUG SCREENING; DRUG SYNTHESIS; ENZYME INHIBITION; HEART; KIDNEY; LUNG; METHODOLOGY; RABBIT; STRUCTURE ACTIVITY RELATION; THEORETICAL STUDY;

ANIMALS; CATTLE; CYCLIC AMP; KIDNEY; KINETICS; LUNG; MYOCARDIUM; PHOSPHODIESTERASE INHIBITORS; PYRAZOLES; PYRIMIDINES; RABBITS;

EID: 0016158566     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00252a016     Document Type: Article

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