Synthetic Thyrotropin-Releasing Factor Analogs. 3.1, 2 Effect of Replacement or Modification of Histidine Residue on Biological Activity

Journal of Medicinal Chemistry

Volumn 15, Issue 5, 1972, Pages 479-482

  Rivier, J ^a   Vale, W ^a   Monahan, M ^a   Ling, N ^a   Burgus, R ^a  

^a SALK INSTITUTE FOR BIOLOGICAL STUDIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACID; HISTIDINE; PEPTIDE; PROTIRELIN;

ANIMAL; ARTICLE; INFRARED RADIATION; MASS SPECTROMETRY; MOUSE; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PROTEIN CONFORMATION; SPECTROSCOPY; STRUCTURE ACTIVITY RELATION; SYNTHESIS; THIN LAYER CHROMATOGRAPHY;

AMINO ACIDS; ANIMAL; CHROMATOGRAPHY, THIN LAYER; HISTIDINE; INFRARED RAYS; MAGNETIC RESONANCE SPECTROSCOPY; MICE; PEPTIDES; PROTEIN CONFORMATION; PROTIRELIN; SPECTRUM ANALYSIS; SPECTRUM ANALYSIS, MASS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0015341526     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00275a010     Document Type: Article

References (24)

1. R. Burgus, T. Dunn, D. M. Desiderio, D. N. Ward, W. Vale, R. Guillemin, A. M. Felix, D. Gillessen, and R. O. Studer, Endocrinology, 86, 573 (1970) (paper 1).
2. W. Vale, J. Rivier, and R. Burgus, Endocrinology, 89, 1485 (1971) (paper 2).
3. K. Hofmann and C. Y. Bowers, J. Med. Chem., 13, 1099 (1970);
4. C. Y. Bowers, A. Weil, J. K. Chang, H. Sievertsson, F. Enzmann, and K. Folkers, Biochem. Biophys. Res. Commun., 60, 683 (1970);
5. J. K. Chang, H. Sievertsson, B. Currie, K. Folkers, and C. Y. Bowers, J. Med. Chem., 14, 484(1971);
6. E. D. Nicolaides, unpublished results;
7. J. F. Wilber and G. Flouret, 53rd Meeting of the Endocrine Society, Abstract 89, June 1971;
8. D. Gillessen, F. Piva, H. Steiner, and R. O. Studer, Heh. Chim. Acta, 54, 1335 (1971).
9. D. Gillessen, A. M. Felix, W. L. Lergier, and R. O. Studer, Heh. Chim. Acta, 54, 236(1970).
10. H. Gibian and E. Klieger. Justus Liebigs Ann. Chem., 640, 145 (1961).
11. J. Biol. Chem., 262, 555 (1967);
12. C. Y. Bowers, A. Weil, J. K. Chang, H. Sievertsson, F. Enzmann, and K. Folkers, Biochem. Biophys. Res. Commun., 40, 683 (1970).
13. P. G. Pietta and G. R. Marshall, Chem. Commun., 650 (1970).
14. F.C. Westall and A. B. Robinson, J. Org. Chem., 35, 2342 (1970).
15. W. Vale, R. Burgus, T. F. Dunn, and R. Guillemin, Hormones, 2, 193 (1970).
16. R. Guillemin, R. Burgus, and W. Vale, Vitam. Horm. (New York), 29, 1 (1971).
17. F. Schneider and W. Schalf, Hoppe Seyler's Z. Physiol. Chem., 327, 74 (1962);
18. J. T. Edsall, “Proteins, Amino Acids, and Peptides,” W. A. Hamor, Ed., Hafner, New York, N. Y., 1943, p 85;
19. F. Schneider, Hoppe Seyler's Z. Physiol. Chem., 336, 26 (1963).
20. M. L. Polan, et al, Biochem. Biophys. Res. Commun., 38, 1127 (1970).
21. E. Stahl, “Thin-layer Chromatography,” E. Stahl, Ed., Academic Press, New York, N. Y., 1965.
22. S. Yamada and H. A. Itano, Biochim. Biophys. Acta, 130, 538 (1966).
23. E. Fischer and L. H. Cone, Justus Liebigs Ann. Chem., 363, 107(1908).
24. V. Bacon, E. Jellum, W. Patton, W. Pereira, and B. Halpern, Biochem. Biophys. Res. Commun., 37, 878 (1969).