Quantification of depletion in solution-type topical preparations in vivo

Journal of Cosmetic Science

Volumn 49, Issue 3, 1998, Pages 165-174

  Leopold, Claudia S ^a  

^a HEINRICH HEINE UNIVERSITY   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0013655162     PISSN: 00379832     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (21)

1. J. L. Zatz, "Percutaneous Absorption: Computer Simulation Using Multicompartmented Membrane Models," in Percutaneous Absorption, R. L. Bronaugh and H. I. Maibach, Eds. (Marcel Dekker, New York, 1985), pp. 165-181.
2. R. H. Guy and J. Hadgraft, A theoretical description relating skin penetration to the thickness of the applied medicament, Int. J. Pharm., 6, 321-332 (1980).
3. E. R. Cooper and B. Berner, Finite dose pharmacokinetics of skin penetration, J. Pharm, Sci., 74, 1100-1102 (1985).
4. J. L. Zatz, Influence of depletion on percutaneous absorption characteristics, J. Soc. Cosmet. Chem., 36, 237-249 (1985).
5. W. J. Addicks, G. Flynn, N. Weiner, and R. Curl, A mathematical model to describe drug release from thin topical applications, Int. J. Pharm., 56, 243-248 (1989).
6. W. Addicks, N. Weiner, G. Flynn, R. Curl, and E. Topp, Topical drug delivery from thin applications: Theoretical predictions and experimental results, Pharm. Res., 7, 1048-1054 (1990).
7. M. Walker, L. A. Chambers, D. A. Hollingsbee, and J. Hadgraft, Significance of vehicle thickness to skin penetration of halcinonide, Int. J. Pharm., 70, 167-172 (1991).
8. G. Levy, Kinetics of pharmacologic effects, Clin. Pharmacol. Ther., 7, 362-371 (1966).
9. B. C. Lippold and H. Reimann, Wirkungsbeeinflussung bei Lösungssalben durch Vehikel am Beispiel von Methylnicotinat, Teil II: Beziehung zwischen relativer thermodynamischer Aktivität und Bioverfügbarkeit: Penetrationsbeschleunigung und Entleerungseffekt, Acta Pharm. Technol., 35, 136-142 (1989).
10. C. S. Leopold and B. C. Lippold, Enhancing effects of lipophilic vehicles on skin penetration of methyl nicotinate in vivo, J. Pharm. Sci., 84, 195-198 (1995).
11. C. S. Leopold and B. C. Lippold, A new application chamber for skin penetration studies in vivo with liquid preparations. Pharm. Res., 9, 1215-1218 (1992).
12. C. S. Leopold, How accurate is the determination of the relative bioavailability of transdermal drug formulations from pharmacodynamic response data? Pharm. Acta Helv., (in press, 1998).
13. B. C. Lippold and H. Reimann, Wirkungsbeeinflussung bei Lösungssalben durch Vehikel am Beispiel von Methylnicotinat, Teil 1: Relative thermodynamische Aktivität des Arzneistoffes in verschiedenen Vehikeln und Freisetzungsverhalten, Acta Pharma. Technol., 35, 128-135 (1989).
14. M. Bach and B. C. Lippold, Penetration enhancement and its quantification, Eur. J. Pharm. Biopharm. (in press, 1998).
15. J. Crank, Mathematics of Diffusion (Oxford University Press, London, 1956).
16. M. Bach and B. C. Lippold, Influence of penetration enhancers on the blanching intensity of betamethasone 17-benzoate, Int. J. Pharm. (in press, 1998).
17. B. J. Aungst, Structure/effect studies of fatty acid isomers as skin penetration enhancers and skin irritants, Pharm. Res., 6, 244-247 (1989).
18. A. H. Ghanem, H. Mahmoud, W. I. Higuchi, P. Liu, and W. R. Good, The effects of ethanol on the transport of lipophilic and polar permeants across hairless mouse skin: Methods/validation of a novel approach, Int. J. Pharm., 78, 137-156 (1992).
19. R. Kadir, D. Stempler, Z. Liron, and S. Cohen, Penetration of adenosine into excised human skin from binary vehicles: The enhancement factor, J. Pharm. Sci. 77, 409-413 (1988).
20. M. Goodman and B. W. Barry, Action of penetration enhancers on human skin as assessed by the permeation of model drugs 5-fluorouracil and estradiol. I. Infinite dose technique, J. Invest. Dermatol., 91, 323-327 (1988).
21. C. S. Leopold and B. C. Lippold, An attempt to clarify the mechanism of the penetration enhancing effects of lipophilic vehicles with differential scanning calorimetry (DSC), J. Pharm. Pharmacol., 47, 276-281 (1995).