[23]Intracellular receptor characterization and ligand screening by transactivation and hormone-binding assays

Methods in Molecular Genetics

Volumn 8, Issue C, 1996, Pages 405-420

  Allegretto, Elizabeth A ^a   Heyman, Richard A ^a  

^a LIGAND PHARMACEUTICALS INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0013574031     PISSN: 10672389     EISSN: None     Source Type: Book Series    
DOI: 10.1016/S1067-2389(96)80056-2     Document Type: Article

References (54)

1. Toft D., and Gorski J. Proc. Natl. Acad. Sci. U.S.A. 55 (1966) 1574
2. Jensen E.V., Hurst D.J., DeSombre E.R., and Jungblut P.W. Science 158 (1967) 385
3. Gardner R.S., and Tomkins G.M. J. Biol. Chem. 244 (1969) 4761
4. Spelsberg T.C., Steggles A.W., and O'Malley B.W. J. Biol. Chem. 246 (1971) 4188
5. Brumbaugh P.F., and Haussler M.R. J. Biol. Chem. 249 (1974) 1258
6. Hollenberg S.M., Weinberger C., Ong E.S., Cerelli G., Oro A., Lebo R., Thompson E.B., Rosenfeld M.G., and Evans R.M. Nature (London) 318 (1985) 635
7. Walter P., Green S., Greene G., Krust A., Bornert J., Jeltsch J., Staub A., Jensen E., Scrace G., Waterfield M., and Chambon P. Proc. Natl. Acad. Sci. U.S.A. 82 (1985) 7889
8. Conneely O.M., Sullivan W.P., Toft D.O., Birnbaumer M., Cook R.G., Maxwell B.L., Zarucki-Schulz T., Greene G.L., Schrader W.T., and O'Malley B.W. Science 233 (1986) 767
9. Jeltsch J.M., Krozowski Z., Quirin-Stricker C., Gronemeyer H., Simpson R.J., Garnier J.M., Krust A., Jacob F., and Chambon P. Proc. Natl. Acad. Sci. U.S.A. 83 (1986) 5424
10. McDonnell D.P., Mangelsdorf D.J., Pike J.W., Haussler M.R., and O'Malley B.W. Science 235 (1987) 1214
11. Giguere V., Ong E.S., Segui P., and Evans R.M. Nature (London) 330 (1987) 624
12. Mangelsdorf D.J., Ong E.S., Dyck J.A., and Evans R.M. Nature (London) 345 (1990) 224
13. Milgrom E., and Bavlieu E.E. Biochim. Biophys. Acta 194 (1969) 602
14. Santi D.V., Sibley C.H., Perriard E.R., Tomkins G.M., and Baxter J.D. Biochemistry 12 (1973) 2412
15. Williams D., and Gorski J. Biochemistry 13 (1974) 5537
16. Scatchard G. Ann. N.Y. Acad. Sci. 51 (1949) 660
17. Evans R.M. Science 240 (1988) 889
18. Trusse M., and Beato M. Endocr. Rev. 14 (1993) 459
19. Umesono K., and Evans R.M. Cell 57 (1989) 1139
20. Gorman C.M., Moffat L.F., and Howard B.H. Mol. Cell. Biol. 2 (1982) 1044
21. Chandler V.L., Maler B.A., and Yamamoto K.R. Cell 33 (1983) 489
22. Giguere V., Hollenberg S.M., Rosenfeld M.G., and Evans R.M. Cell 46 (1986) 645
23. Mangelsdorf D.J., Umesono K., and Evans R.M. In: Sporn M., Roberts A.B., and Goodman D.S. (Eds). The Retinoids: Biology, Chemistry, and Medicine (1994), Raven Press, Cold Spring Harbor, New York 319
24. Berger T.S., Parandoosh Z., Perry B.W., and Stein R.B. J. Steroid Biochem. 41 (1992) 733
25. Wigler M., Sweet R., Sim G.K., Wold B., Pellicer A., Lacy E., Maniatis T., Silverstein S., and Axel R. Cell 16 (1979) 777
26. Petkovitch M., Brand N.J., Krust A., and Chambon P. Nature (London) 330 (1987) 444
27. Levin A.A., Sturzenbecker L.J., Kazmer S., Bosakowski T., Huselton C., Allenby G., Speck J., Kratzeisen C.I., Rosenberger M., Lovey A., and Grippo J.F. Nature (London) 355 (1992) 359
28. Heyman R.A., Mangelsdorf D.J., Dyck J.A., Stein R.B., Eichele G., Evans R.M., and Thaller C. Cell 68 (1992) 397
29. Allegretto E.A., McClurg M.R., Lazarchik S.B., Clemm D.L., Kerner S.A., Elgort M.G., Boehm M.F., White S.K., Pike J.W., and Heyman R.A. J. Biol. Chem. 268 (1993) 26625
30. Lotan R. Biochim. Biophys. Acta 605 (1980) 33
31. Allegretto E.A., Kelley M.A., Donaldson C.A., Levine N., Pike J.W., and Haussler M.R. Biochem. Biophys. Res. Commun. 116 (1983) 75
32. Yang N., Schule R., Mangelsdorf D.J., and Evans R.M. Proc. Natl. Acad. Sci. U.S.A. 88 (1991) 3559
33. Keidel S., Rupp E., and Szardenings M. Eur. J. Biochem. 204 (1992) 1141
34. Allenby G., Bocquel M.T., Saunders M., Kazmer S., Speck T., Rosenberger M., Lovey A., Kastner P., Grippo J.F., Chambon P., and Levin A.A. Proc. Natl. Acad. Sci. U.S.A. 90 (1993) 30
35. Boehm M.F., McClurg M.R., Pathirana C., Mangelsdorf D.J., White S.K., Hebert J., Winn D., Goldman M.E., and Heyman R.A. J. Med. Chem. 37 (1994) 408
36. Benbrook D., Lernhardt E., and Pfahl M. Nature (London) 333 (1988) 669
37. Ishikawa T., Umesono K., Mangelsdorf D.J., Aburtani H., Stanger V.Z., Shibasaki Y., Imaware M., Evans R.M., and Takaku F. Mol. Endocrinol. 4 (1990) 837
38. Mangelsdorf D.J., Borgmeyer U., Heyman R.A., Zhou J.Y., Ong E.S., Oro A.E., Kakizuka A., and Evans R.M. Genes Dev. 6 (1992) 329
39. Burnside J., Darling D.S., and Chin W.W. J. Biol. Chem. 265 (1990) 2500
40. Sone T., Ozona K., and Pike J.W. Mol. Endocrinol. 5 (1991) 1578
41. Yu V.C., Delsert C., Andersen B., Holloway J.M., Devary O., Naar A.M., Kim S.Y., Boutin J., Glass C.K., and Rosenfeld M.G. Cell 67 (1991) 1251
42. Zhang X., Hoffmann B., Tran P., Graupner G., and Pfahl M. Nature (London) 355 (1992) 441
43. Leid M., Kastner P., Lyons R., Nakshatri H., Saunders M., Zacharewski T., Chen J., Staub A., Garniert J., Mader S., and Chambon P. Cell 68 (1992) 377
44. Kliewer S.A., Umesono K., Mangelsdorf D.J., and Evans R.M. Nature (London) 355 (1992) 446
45. McDonnell D.P., Pike J.W., Drutz D.J., Butt T.R., and O'Malley B.W. Mol. Cell. Biol. 9 (1989) 3517
46. McDonnell D.P., Nawaz Z., Densmore C., Weigel N.L., Pham T.A., Clark J.H., and O'Malley B.W. J. Steroid Biochem. Mol. Biol. 39 (1991) 291
47. Metzger D., White J.H., and Chambon P. Nature (London) 334 (1988) 31
48. Schena M., and Yamamoto K.R. Science 241 (1988) 965
49. Mangelsdorf D.J., Umesono K., Kliewer S.A., Borgmeyer U., Ong E.S., and Evans R.M. Cell 66 (1991) 555
50. Sucov H.M., Murakami K.K., and Evans R.M. Proc. Natl. Acad. Sci. U.S.A. 87 (1990) 5392
51. Hoffmann B., Lehmann J.M., Zhang X., Hermann T., Husmann M., Graupner G., and Pfahl M. Mol. Endocrinol. 4 (1990) 1727
52. de Thé H., Vivanco-Ruiz M.M., Tiollais P., Stunnenberg H., and Dejean A. Nature (London) 343 (1990) 177
53. Heery D.M., Zacharewski T., Pierrat B., Gronemeyer H., Chambon P., and Losson R. Proc. Natl. Acad. Sci. U.S.A. 90 (1993) 4281
54. Hall B.L., Smit-McBride Z., and Privalsky M. Proc. Natl. Acad. Sci. U.S.A. 90 (1993) 6929