Versatile solid-phase synthesis of S-arylisothioureas

Journal of Combinatorial Chemistry

Volumn 4, Issue 4, 2002, Pages 290-294

  Katritzky, Alan R ^a   Rogovoy, Boris V ^a   Vvedensky, Vladimir ^a   Kovalenko, Katherine ^a   Forood, Behrouz ^b  

^a University of Florida ^*  (United States)

^b Cypress Bioscience Inc   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ARTICLE;

EID: 0012462001     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc010065d     Document Type: Article

References (14)

1. Zhang. J.; McCarthy, T. J.; Moore, W. M.; Currie, M. G.; Welch, M. J. J. Med. Chem. 1996, 39, 5110.
2. Wei, L. H.; Arabolos, N.; Ignarro, L. J. Nitric Oxide 1998, 2, 155.
3. Cooper, G. R.; Mialkowski, K.; Wolff, D. J. Arch. Biochem. Biophys. 2000, 375, 183.
4. Southan, G. J.; Gauld, D.; Lubeskie, A.; Zingarelli, B.; Cuzzocrea, S.; Salzman, A. L.; Szabo, C.; Wolff, D. J. Biochem. Pharmacol. 1997, 54, 409.
5. Mertens, A.; Koenig, B.; Leser, U. Preparation of (thio)-carbamidinic acid derivatives from isothioureas and (thio)-isocyanates for antiviral pharmaceuticals. Int. Pat. WO 95/ 04034, 1995. (Chem. Abstr. 1995, 122. 265045).
6. Pascual, A.; Rindlisbacher, A. Pestic. Sci. 1994, 42, 253
7. Kogan, M.; Dinizo, S. E.; Fancher, L. W. Preparation of herbicidal N,N′-(N″-isopropylcarbamoyl,N‴-isopropylcarbamoyl)-S- ethylisothiourea. U.S. Patent 4,714,493, 1987. (Chem. Abstr. 1987, 107, 111110).
8. Booth, S.; Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1997, 53, 5643.
9. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1998, 54, 15385.
10. Katritzky, A. R.; Rogovoy, B. V.; Chassaing, C.; Vvedensky, V. Y. J. Org. Chem. 2000, 65, 8080.
11. (a) Ngu, K.; Patel, D. V. Tetrahedron Lett. 1997, 38, 973.
12. (b) Mjalli, A. M. M.; Toyonaga, B. E. In Molecular Diversity and Combinatorial Chemistry: Libraries and Drug Discovery; Chaiken, I. M., Janda, K. D., Eds.: American Chemical Society: Washington, DC, 1996; p 70.
13. Fivush, A. M.; Willson, T. M. Tetrahedron Lett. 1997, 38, 7151.
14. Shtefan, E. D.; Vvedenskii, V. Y. Russ. Chem. Rev. 1996, 65, 307-314.