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Volumn 639, Issue , 1996, Pages 228-243

Syntheses, Biological Activity, and Conformational Analysis of Fluorine-Containing Taxoids

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EID: 0012077542     PISSN: 00976156     EISSN: None     Source Type: Book Series    
DOI: None     Document Type: Article
Times cited : (22)

References (63)
  • 2
    • 77956791953 scopus 로고
    • J. A. Bristol, Ed.; Academic Press: San Diego, Chapter 32
    • Suffness, M. In Annual Reports in Medicinal Chemistry; J. A. Bristol, Ed.; Academic Press: San Diego, 1993; Vol. 28; Chapter 32, pp 305-314.
    • (1993) Annual Reports in Medicinal Chemistry , vol.28 , pp. 305-314
    • Suffness, M.1
  • 13
    • 85083127376 scopus 로고    scopus 로고
    • Georg, G. I., 3′-N-(4-Azido-2,3,5,6-tetrafluorobenzoyl)paclitaxel and 7-(4-Azido-2,3,5,6-tetrafluorobenzoyl)paclitaxel have been synthesized as potential photoaffinity labels. See Ref. 14
    • Georg, G. I., 3′-N-(4-Azido-2,3,5,6-tetrafluorobenzoyl)paclitaxel and 7-(4-Azido-2,3,5,6-tetrafluorobenzoyl)paclitaxel have been synthesized as potential photoaffinity labels. See Ref. 14.
  • 15
    • 85083146035 scopus 로고    scopus 로고
    • Chen, S.-H., For the incorporation of fluorine to the baccatin moiety, see Refs. 16 and 17
    • Chen, S.-H., For the incorporation of fluorine to the baccatin moiety, see Refs. 16 and 17.
  • 17
    • 0001843250 scopus 로고
    • Taxane Anticancer Agents: Basic Science and Current Status
    • G. I. Georg; T. T. Chen; I. Ojima and D. M. Vyas, Ed.; American Chemical Society: Washington D.C.
    • Chen, S. H.; Farina, V. In Taxane Anticancer Agents: Basic Science and Current Status; G. I. Georg; T. T. Chen; I. Ojima and D. M. Vyas, Ed.; ACS Symp. Series 583; American Chemical Society: Washington D.C., 1995; pp 247-261.
    • (1995) ACS Symp. Series 583 , pp. 247-261
    • Chen, S.H.1    Farina, V.2
  • 20
    • 0002439670 scopus 로고
    • Taxane Anticancer Agents: Basic Science and Current Status
    • G. I. Georg; T. T. Chen; I. Ojima and D. M. Vyas, Ed.; American Chemical Society: Washington D. C.
    • Vuilhorgne, M.; Gaillard, C.; Sanderlink, G. J.; Royer, I.; Monsarrat, B.; Dubois, J.; Wright, M. In Taxane Anticancer Agents: Basic Science and Current Status, G. I. Georg; T. T. Chen; I. Ojima and D. M. Vyas, Ed.; ACS Symp. Series 583; American Chemical Society: Washington D. C., 1995; pp 98-110.
    • (1995) ACS Symp. Series 583 , pp. 98-110
    • Vuilhorgne, M.1    Gaillard, C.2    Sanderlink, G.J.3    Royer, I.4    Monsarrat, B.5    Dubois, J.6    Wright, M.7
  • 25
    • 85083149002 scopus 로고    scopus 로고
    • 50(paclitaxel) = 1.2
    • 50(paclitaxel) = 1.2.
  • 27
    • 85083127330 scopus 로고    scopus 로고
    • 50(docetaxel) = 1.49; %T/C = 6; log cell kill 3.2) (see Ref. 28)
    • 50(docetaxel) = 1.49; %T/C = 6; log cell kill 3.2) (see Ref. 28).
  • 30
    • 0002511289 scopus 로고
    • A. Hassner, Ed.; JAI Press: Greenwich
    • Ojima, I. In Advances in Asymmetric Synthesis; A. Hassner, Ed.; JAI Press: Greenwich, 1995; Vol. 1; pp 95-146.
    • (1995) Advances in Asymmetric Synthesis , vol.1 , pp. 95-146
    • Ojima, I.1
  • 57
    • 85083127120 scopus 로고    scopus 로고
    • Georg, G. I., For a comprehensive review on the conformational studies on paclitaxel and docetaxel, see Ref. 58
    • Georg, G. I., For a comprehensive review on the conformational studies on paclitaxel and docetaxel, see Ref. 58.
  • 61
    • 85083120678 scopus 로고    scopus 로고
    • 2O (3:1) could be perfomed at -20 °C (see Ref. 18), but we did not have any luck in keeping the solution from freezing below 0 °C although we were able to obtain clean NMR spectra in glassy state at -20 °C
    • 2O (3:1) could be perfomed at -20 °C (see Ref. 18), but we did not have any luck in keeping the solution from freezing below 0 °C although we were able to obtain clean NMR spectra in glassy state at -20 °C.
  • 63
    • 85083120922 scopus 로고    scopus 로고
    • Ojima, I.; Kuduk, S. D.; Chakravarty, S.; Ourevitch, M., Unpublished results
    • Ojima, I.; Kuduk, S. D.; Chakravarty, S.; Ourevitch, M., Unpublished results.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.