2-sulfinyl benzothiazoles, -oxazoles and -imidazoles are novel in vitro bone anti-reabsorptive compounds

Medicinal Chemistry Research

Volumn 7, Issue 3, 1997, Pages 151-167

  Corbett, J W ^a   Kerr, J S ^a   Wong, P ^a   Harlow, P ^a   Boswell, G A ^a   Pease, L ^b   Lee, B S ^c   Holliday, L S ^c   Gluck, S L ^c  

^a DUPONT COMPANY   (United States)

^b ABBOTT LABORATORIES   (United States)

^c WASHINGTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0010264252     PISSN: 10542523     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (40)

1. Forgac, M. Physiol. Rev., 1989, 69, 765.
2. Palokangasm, H.; Metsikkö, K.; Väänänen, K. J. Biol. Chem., 1994, 269, 17577.
3. Vaes, G. Clin. Orthoped. Related Res., 1988, 231, 239.
4. Blair, H.C.; Kahn, J.; Crouch, E.C.; Jeffrey, J.J.; Teitelbaum, S.L. J. Cell Biol., 1986, 102, 1164.
5. Gluck, S.L. J. Bioenerg. Biomembr., 1992, 24, 354.
6. Xie, X.-S.; Crider, B.P.; Ma, Y.-M.; Stone, D.K. J. Biol. Chem., 1994, 269, 25809.
7. Nelson, N. J. Bioenerg. Biomembr., 1989, 21, 553.
8. Peng, S.-B.; Zhang, Y.; Crider, B.P.; White, A.E.; Fried, V.A.; Stone, D.K.; Xie, X.-S. J. Biol. Chem., 1994, 269, 27778.
9. Nelson, N. Current Opinion in Cell Biology, 1994, 4, 654.
10. Gluck, S.L. Int. Rev. Cytol., 1993, 137C, 105.
11. Chatterjee, D.; Chakraborty, M.; Leit, M.; Neff, L.; Jamsa-Kellokumpu, S.; Fuchs, R.; Baron, R. Proc. Natl. Acad. Sci. USA , 1992, 89, 6257.
12. Crider, B.P.; Xie, X.-S.; Stone, D.K. J. Biol. Chem., 1994, 269, 17379.
13. Werner, G.; Hagenmaier, H. J. Antibiot., 1984, 37, 110.
14. Baron, R.; Chakraborty, M.; Chatterjee, D.; Horne, W.; Lomri, A.; Ravesloot, J.-H. Handbook of Experimental Pharmacology, 1993, 3, 111.
15. Feng, Y.; Forgac, M. J. Biol. Chem., 1994, 269, 13224.
16. Feng, Y.; Forgac, M. J. Biol. Chem., 1992, 267, 5817.
17. Lindberg, P.; Wallmark, B.; Väänänen, K.; Håkanson, R. Patent application WO8903829, 1989.
18. Lindberg, P.; Brändström, A.; Wallmark, B.; Mattsson, H.; Rikner, L.; Hoffmann, K.-J. Med. Res. Rev., 1990, 10, 1.
19. Mizunashi, K.; Furukawa, Y.; Katano, K.; Abe, K. Calcif. Tissue Int., 1993, 53, 21.
20. David, P.; Home, W.C.; Baron, R. Biochem. Biophys. Acta, 1996, 1280, 155.
21. Hall, T.J.; Schaueblin, M. J. Bone Miner. Res., 1994, 27, 159.
22. Sundquist, K.; Lakkakorpi, P.; Wallmark, B.; Väänänen, K. Biochem. Biophys. Res. Commun., 1990, 168, 309.
23. Mattsson, J.P.; Väänänen, K.; Wallmark, B.; Lorentzon, P. Biochem. Biophys. Acta., 1991, 1065, 261.
24. Tuukanen, J.; Väänänen, H.K. Calcif. Tissue Int., 1986, 38, 123.
25. Santilli, A.A.; Scotese, A.C.; Strike, D.P. Patent application EP 434405 A1, 1990.
26. Bex, F.J.; Santilli, A.A.; Kees, K. Cur. Opin. Invest. Drugs, 1993, 2, 397.
27. Santilli, A.A.; Bex, F.J. Curr. Opin. Ther., 1993, 3, 23.
28. Gluck, S.; Al-Awqati, A. J. Clin. Invest., 1984, 73, 1704.
29. Gluck, S.; Caldwell, J. J. Biol. Chem., 1987, 262, 15780.
30. Holliday, L.S.; Dean, A.D.; Greenwald, J.E.; Gluck, S.L. J. Biol. Chem., 1995, 270, 1.
31. Lerner, U.H.; Ransjoe, M.; Ljunggren, O.; Klaushofer, K.; Hoffmann, O.; Peterlik, M. J. Bone Miner. Res., 1991, 6, 551.
32. Lerner, U.H. J. Bone Miner. Res., 1987, 2, 375.
33. Lerner, U.H.; Ohlin, A. J. Bone Miner. Res., 1993, 8, 147.
34. Takahashi, N.; Akatsu, T.; Sasaki, T.; Nicholson, G.C.; Moseley, J.M.; Martin, T.J.; Suda, T. Endocrinology, 1988, 123, 1504.
35. Wang, Z.-Q.; Hemken, P.; Menton, D.; Gluck, S. Am. Physiol. Soc., 1992, 263, F277.
36. Blair, H.C.; Teitelbaum, S.L.; Ghiselli, R.; Gluck, S. Science, 1989, 245, 855.
37. Still, W.C.; Kahn, M.; Mitra, A. J. Org. Chem., 1978, 43, 2923.
38. Fabricant, C.; David, P.; Chatterjee, D.; Baron, R. J. Bone Miner. Res., 1993, 8, S392.
39. Fiorentino, M.; Testaferri, L.; Tiecco, M.; Troisi L.J. Chem. Soc., Chem. Commun., 1997, 316.
40. Lorin C.; Marot, C.; Rollin , P. Tetrahedron Lett., 1995, 36, 4437.