1,3-Diarylpyrazolo[4,5-c]- and -[5,4-c]quinolin-4-ones. 4. Synthesis and Specific Inhibition of Benzodiazepine Receptor Binding

Journal of Medicinal Chemistry

Volumn 30, Issue 10, 1987, Pages 1737-1742

  Palazzino, Giovanna ^a   Cecchi, Lucia ^a   Melani, Fabrizio ^a   Colotta, Vittoria ^a   Filacchioni, Guido ^a   Martini, Claudia ^b   Lucacchini, Antonio ^b  

^a UNIVERSITY OF FLORENCE   (Italy)

^b UNIVERSITY OF PISA   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

BENZODIAZEPINE RECEPTOR; CHLORDIAZEPOXIDE; DIAZEPAM; FLUNITRAZEPAM H 3; PYRAZOLO[4,5 C]QUINOLIN 4 ONE DERIVATIVE; PYRAZOLO[5,4 C]QUINOLIN 4 ONE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SYNTHESIS; NONHUMAN;

ANIMAL; BINDING, COMPETITIVE; BRAIN; CATTLE; FLUNITRAZEPAM; ISOMERISM; MAGNETIC RESONANCE SPECTROSCOPY; MEMBRANES; PYRAZOLES; QUINOLINES; RECEPTORS, GABA-A; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0005175003     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00393a009     Document Type: Article

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