A new efficient synthesis of ω-aminoalkylidene-1,1-bisphosphonate tetraethylesters

Phosphorus, Sulfur and Silicon and Related Elements

Volumn 132, Issue , 1998, Pages 219-229

  Gourves, Jean Philippe ^a   Couthon, Hélène ^a   Sturtz, Georges ^a  

^a UNIVERSITÉ DE BRETAGNE OCCIDENTALE   (France)

Author keywords

Amination; Methylidenebisphosphonate; Tetraethyl aminoalkylidenebisphosphonates and hydroxy alkylidenebisphosphonates

Indexed keywords

EID: 0002329425     PISSN: 10426507     EISSN: None     Source Type: Journal    
DOI: 10.1080/10426509808036988     Document Type: Article

References (20)

1. O.L.M. BIJVOET, H.A. FLEISCH, R.E. CANFIELD, R.G.G. RUSSELL (eds.), « Bisphosphonates on bones » © Elsevier Science B.V. (1995).
2. D.K.J. HOSKING, Drugs, 40, 829-840 (1990).
3. H. FLEISCH, Drugs, 42, 919-944 (1991).
4. S.E. PAPAPLOULOS, J.O. LANOMAN, O.L.M. BIJVOET, C.W.G.M LOWIX, R. VALKEMA, E.K.J. PAUWELS, P. VERMEIJ, Bone, 13, S41-S49 (1992).
5. a - G. STURTZ, G. APPERE, K. BREISTOL, O. FOSTAD, G. SCHWARTSMANN, H.R. HENDRIKS, Eur. J. Med. Chem., 27, 825-833 (1993)
6. b - G. STURTZ, H. COUTHON, O. FABULET, M. MIAN, S. ROSINI, Eur. J. Med. Chem., 28, 899-903 (1993)
7. c - F. HOSAIN, R.P. SPENCER, H.M. COUTHON, G.L. STURTZ, J. Nucl. Med. 37, 105-107 (1996).
8. L. MAIER, Phosphorus and Sulfur, 11, 311-322 (1981).
9. G. STURTZ, H. COUTHON, C. R. Acad. Sci. Paris, t 316, série II, 181-186 (1993).
10. G. APPERE, Ph. D. Thesis, 1990, U.B.O. Brest.
11. T. BAILLY, R. BURGADA, Phosphorus, Sulfur and Silicon, 86, 217-228 (1994).
12. O.E.O. HORMI, E.O. PAJUNEN, A.K.C. AVALL, P. PENNAMEN, Synth. Comm., 20, 1865-1867 (1990).
13. E. BOSIES, A. ESSWEIN, F. BAUSS, Ger. Offen. DE 4,029,499 [CA 116-P23596ls].
14. H. BIERE, C. RUFER, I. BOETTCHER, Ger Offen. DE 3,225,469 [CA 100-P210141f].
15. D.W. HUTCHINSON, D.M. THORNTON, Synthesis, 135-137 (1990).
16. A. BONGINI, G. CARDILLO, M. ONENA, Synthesis, 618-620 (1979).
17. st ed. 2, 308-310 (1995).
18. H. STAUDINGER, J. MEYER, Helv. Chim. Acta. 2, 635-646 (1919).
19. N. KNOUZI, M. VAULTIER, R. CARRIE, Bull. Soc. Chim. Fr., (5), 815-819 (1985).
20. G. STURTZ, A. PONDAVEN-RAPHALEN, Phosphorus and Sulfur, 36, 39-52A (1988).