Biginelli condensations of fluorinated 3-oxo esters and 1,3-diketones

Journal of Fluorine Chemistry

Volumn 103, Issue 1, 2000, Pages 17-23

  Saloutin, V I ^a   Burgart, Ya V ^a   Kuzueva, O G ^a   Kappe, C O ^b   Chupakhin, O N ^a  

^a INSTITUTE OF ORGANIC SYNTHESIS   (Russian Federation)

^b UNIVERSITY OF GRAZ   (Austria)

Author keywords

Biginelli reaction; Fluoroalkyl 3 oxo esters and 1,3 diketones; Hexahydropyrimidines

Indexed keywords

EID: 0002035865     PISSN: 00221139     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0022-1139(99)00216-X     Document Type: Article

References (15)

1. Synthesis and reactions of biginelli compounds, part 18. For part 17, see: C.O. Kappe, Bioorg. Med. Chem. Lett. in press.
2. Synthesis and reactions of biginelli compounds, part 18. For part 17, see: C.O. Kappe, Bioorg. Med. Chem. Lett. in press.
3. C.O. Kappe, Synthesis (1999) 1799.
4. C.O. Kappe, D. Kumar, R.S. Varma, Synthesis (1999), in press.
5. Kappe C.O., Falsone S.F., Fabian W.M.F., Belaj F. Heterocycles. 51:1999;77.
6. A.M. Lovelace, D.A. Rausch, M. Postelnek, Aliphatic Fluorine-Containing Compounds, Inostrannaya Literatura, Moscow, 1961, p. 225.
7. Henne A.L., Newman M.S., Quill L.L., Staniforth R.A. J. Amer. Chem. Soc. 69:1947;1819.
8. Akhtar M.S., Seth M., Bhaduri A.P. Indian J. Chem. 26B:1987;556.
9. G.C. Levy, R.L. Lichter, G.L. Nelson, Carbon-13 Nuclear Magnetic Resonance Spectroscopy, Wiley, New York, 1980, p. 338.
10. Pashkevich K.I., Saloutin V.I., Postovskii I.Y. Russ. Chem. Rev. 50:1981;325.
11. Kappe C.O. J. Org. Chem. 62:1997;7201.
12. K.I. Pashkevich, Z.E. Skryabina, V.I. Saloutin, Russ. Chem. Bull. (1987) 2527.
13. Skryabina Z.E., Burgart Ya.V., Saloutin V.I. Russ. J. Org. Chem. 33:1997;442.
14. Burgart Ya.V., Fokin A.S., Kuzueva O.G., Chupakhin O.N., Saloutin V.I. J. Fluor. Chem. 92:1998;101.
15. Kappe C.O., Roschger P. J. Heterocycl. Chem. 26:1989;55.