-
6
-
-
0023924162
-
-
(1988) 44:2081-2086.
-
Naik RQ, Kattige SI, Bhat SV, Alrejy B, de Souza NJ, Rupp RH: An antiinflammatory piperidinylbenzopyranone from Dysoxylum binectariterurrr. isolation, structure and total synthesis. Tetrahedron (1988) 44:2081-2086.
-
Kattige SI, Bhat SV, Alrejy B, de Souza NJ, Rupp RH: An Antiinflammatory Piperidinylbenzopyranone from Dysoxylum Binectariterurrr. Isolation, Structure and Total Synthesis. Tetrahedron
-
-
Naik, R.Q.1
-
8
-
-
0029807115
-
-
ofcyclins.
-
Sedlacek HH, Czech J, Naik R, Kaur G, Worland P, Losiewicz M: Flavopiridol L86-8275, NSC-S49890), a new kinase inhibitor for tumor-therapy. Inter J Oncology (1996) 9:1143-1168. A comprehensive review of the preclinical pharmacology of llavopiridol and a review of the role ofcyclins.
-
Czech J, Naik R, Kaur G, Worland P, Losiewicz M: Flavopiridol L86-8275, NSC-S49890, A New Kinase Inhibitor for Tumor-therapy. Inter J Oncology (1996) 9:1143-1168. A Comprehensive Review of the Preclinical Pharmacology of Llavopiridol and A Review of the Role
-
-
Sedlacek, H.H.1
-
11
-
-
0031019034
-
-
cells.
-
Drees M, Dengler WA, Roih T, Labonte H, Mayo J, Malspeis L, Grever M, Sausville EA, Fiebig HH: Flavopiridol (L868275): sélective antitumor activity In vitro. Clinical Cancer Research (1997) 3:273-279. Results demonstrate flavoplridol's selective actions on particular tumor cells.
-
Dengler WA, Roih T, Labonte H, Mayo J, Malspeis L, Grever M, Sausville EA, Fiebig HH: Flavopiridol (L868275): Sélective Antitumor Activity in Vitro. Clinical Cancer Research (1997) 3:273-279. Results Demonstrate Flavoplridol's Selective Actions on Particular Tumor
-
-
Drees, M.1
-
12
-
-
0031963058
-
-
(1998) 91:458-465.
-
Parker BW, Kaur G, Nieves-Neira W, Taimi M, Kohlhagen G, Shimizu T, Losiewicz MD, Pommier Y, Sausville EA, Senderowicz AM: Early Induction of apoptosis in hematopoietic cell lines after exposure to flavopiridol. Blood (1998) 91:458-465.
-
Kaur G, Nieves-Neira W, Taimi M, Kohlhagen G, Shimizu T, Losiewicz MD, Pommier Y, Sausville EA, Senderowicz AM: Early Induction of Apoptosis in Hematopoietic Cell Lines after Exposure to Flavopiridol. Blood
-
-
Parker, B.W.1
-
19
-
-
0030933050
-
-
vitro.
-
Medina JH, Viola H, Wolfman C, Marder M, Wasowski C, Calvo D, Paladini AC: Flavonoids: a new family of benzodiazepine receptor ligands. Neurochem Res (1997) 22:419-425. A short review of a new class of agents with a selective effect on benzodiazepine receptors in vivo and in vitro.
-
Viola H, Wolfman C, Marder M, Wasowski C, Calvo D, Paladini AC: Flavonoids: A New Family of Benzodiazepine Receptor Ligands. Neurochem Res (1997) 22:419-425. A Short Review of A New Class of Agents with A Selective Effect on Benzodiazepine Receptors in Vivo and in
-
-
Medina, J.H.1
-
20
-
-
0025136261
-
-
(1990) 40:2227-2231.
-
Medina JH, Paladini AC, Wolfman C, Levi de Stein M, Calvo D, Diaz L: Chrysin (5,7-dihydroxyflavone), a naturally-occuring ligand for benzodiazepine receptors, with anticonvulsant properties. Biochem Pharmacol (1990) 40:2227-2231.
-
Paladini AC, Wolfman C, Levi de Stein M, Calvo D, Diaz L: Chrysin (5,7-dihydroxyflavone), A Naturally-occuring Ligand for Benzodiazepine Receptors, with Anticonvulsant Properties. Biochem Pharmacol
-
-
Medina, J.H.1
-
21
-
-
0000593328
-
-
receptors. Phytomedicine(1996) 3:29-31.
-
Marder M, Viola H, Wasowski C, Wolfman C, Waterman PG, Medina JH, Paladini AC: Cirsiliol and caffeic acid ethyl ester, isolated from Salvia guaranitica, are competitive ligands for the central benzodiazepine receptors. Phytomedicine(1996) 3:29-31.
-
Viola H, Wasowski C, Wolfman C, Waterman PG, Medina JH, Paladini AC: Cirsiliol and Caffeic Acid Ethyl Ester, Isolated from Salvia Guaranitica, Are Competitive Ligands for the Central Benzodiazepine
-
-
Marder, M.1
-
22
-
-
33746556223
-
-
Wrigley S, Hayes M, Thomas R, Chrystal E (Eds), Royal Society of Chemistry, Cambridge, (1997):30-40. A brief review of the experience of Xenova on screening natural products from different sources.
-
Chicarelli-Robinson Ml, Gibbons S, McNicholas C, Robinson N, Moore M, Faulh U, Wrigley SK: Plants and microbes as complementary sources of chemical diversity for drug discovery. In: Phytochemical Diversity. A Source of New Industrial Products, Wrigley S, Hayes M, Thomas R, Chrystal E (Eds), Royal Society of Chemistry, Cambridge, (1997):30-40. A brief review of the experience of Xenova on screening natural products from different sources.
-
Gibbons S, McNicholas C, Robinson N, Moore M, Faulh U, Wrigley SK: Plants and Microbes As Complementary Sources of Chemical Diversity for Drug Discovery. In: Phytochemical Diversity. A Source of New Industrial Products
-
-
Ml, C.-R.1
-
23
-
-
0028792457
-
-
effects.
-
Marder M, Viola H, Wasowski C, Wolfman C, Waterman PG, Medina JH, Paladini AC: 6,3′-Dinitroflavone, a novel high affinity ligand for the benzodiazepine receptor with potent anxiolytic properties. Bioorg Med Chem Letters (1995) 5:2717-2720. Results indicate very high activity in vivo, with few sedative or muscle relaxant effects.
-
Viola H, Wasowski C, Wolfman C, Waterman PG, Medina JH, Paladini AC: 6,3′-Dinitroflavone, A Novel High Affinity Ligand for the Benzodiazepine Receptor with Potent Anxiolytic Properties. Bioorg Med Chem Letters (1995) 5:2717-2720. Results Indicate Very High Activity in Vivo, with Few Sedative or Muscle Relaxant
-
-
Marder, M.1
-
24
-
-
0004396593
-
-
(1996) 223:384-389.
-
Marder M, Viola H, Wasowski C, Wolfman C, Waterman PG, Cassels BK, Medina JH, Paladini AC: 6-Bromoflavone, a high affinity ligand for the central benzidiazepine receptor is a member of a family of active flavonoids. Biochem Biophys Res Comm (1996) 223:384-389.
-
Viola H, Wasowski C, Wolfman C, Waterman PG, Cassels BK, Medina JH, Paladini AC: 6-Bromoflavone, A High Affinity Ligand for the Central Benzidiazepine Receptor Is A Member of A Family of Active Flavonoids. Biochem Biophys Res Comm
-
-
Marder, M.1
-
25
-
-
0029150673
-
-
(1995) 48:568-573.
-
Ainsworth AM, Chicarelli-Robinson Ml, Copp BR, Fauth U, Hylands PJ, Holloway JA, Latif M, Obeirne GB, Porter N, Renno DV, Richards M, Robinson N: Xenovulene-A, a novel GABA-benzodiazepine receptor binding compound produced by Acremonium strictum. J Antibiotics (1995) 48:568-573.
-
Chicarelli-Robinson Ml, Copp BR, Fauth U, Hylands PJ, Holloway JA, Latif M, Obeirne GB, Porter N, Renno DV, Richards M, Robinson N: Xenovulene-A, A Novel GABA-benzodiazepine Receptor Binding Compound Produced by Acremonium Strictum. J Antibiotics
-
-
Ainsworth, A.M.1
-
29
-
-
0026647540
-
-
(1992) 35:2736-2743.
-
Kashman Y, Gustafson KR, Fuller RW, Cardellina JH, McMahon JB, Currens MJ, Buckheit RW, Hughes SH, Cragg GM, Boyd MR: HIV inhibitory natural products. 7. The calanolides, a novel HIV-lnhibitory class of coumarin derivatives from the tropical rain-forest tree, Calophyllum lanigerum. J Med Chem (1992) 35:2736-2743.
-
Gustafson KR, Fuller RW, Cardellina JH, McMahon JB, Currens MJ, Buckheit RW, Hughes SH, Cragg GM, Boyd MR: HIV Inhibitory Natural Products. 7. the Calanolides, A Novel HIV-lnhibitory Class of Coumarin Derivatives from the Tropical Rain-forest Tree, Calophyllum Lanigerum. J Med Chem
-
-
Kashman, Y.1
-
30
-
-
0027151862
-
-
(1993)36:1110
-
Kashman Y, Gustafson KR, Fuller RW, Cardellina JH, McMahon JB, Currens MJ, Buckheit RW, Hughes SH, Cragg GM, Boyd MR: Correction: The calanolides, a novel HIV-lnhibitory class of coumarin derivatives from the tropical rain-forest tree, Calophyllum lanigerum. J Med Chem (1993)36:1110
-
Gustafson KR, Fuller RW, Cardellina JH, McMahon JB, Currens MJ, Buckheit RW, Hughes SH, Cragg GM, Boyd MR: Correction: the Calanolides, A Novel HIV-lnhibitory Class of Coumarin Derivatives from the Tropical Rain-forest Tree, Calophyllum Lanigerum. J Med Chem
-
-
Kashman, Y.1
-
31
-
-
0027725169
-
-
(1993)36:4131-4138.
-
Patil AD, Freyer AJ, Eggleston DS, Haltiwanger RC, Bean MF, Taylor PB, Caranfa MJ, Breen AL, Bartus HR, Johnson RK, Hertzberg RP, Westley JW: The inophyllums, novel inhibitors of HIV-1 reverse transcriptase from the Malaysian tree Calophyllum Inophyllum. J Med Chem (1993)36:4131-4138.
-
Freyer AJ, Eggleston DS, Haltiwanger RC, Bean MF, Taylor PB, Caranfa MJ, Breen AL, Bartus HR, Johnson RK, Hertzberg RP, Westley JW: the Inophyllums, Novel Inhibitors of HIV-1 Reverse Transcriptase from the Malaysian Tree Calophyllum Inophyllum. J Med Chem
-
-
Patil, A.D.1
-
33
-
-
33746524468
-
-
Chemistry, Cambridge, (1997):1-29.
-
Cragg GM, Boyd MR, Christini MA, Kneller R, Mays TD, Mazan KD, Newmann DJ, Sausville EA: Screening of natural products of plant, microbial and marine origin. In: Phytochemlcal Diversity. A Source of New Industrial Products. Wrigley S, Hayes M, Thomas R, Chrystal E (Eds), Royal Society of Chemistry, Cambridge, (1997):1-29.
-
Boyd MR, Christini MA, Kneller R, Mays TD, Mazan KD, Newmann DJ, Sausville EA: Screening of Natural Products of Plant, Microbial and Marine Origin. In: Phytochemlcal Diversity. A Source of New Industrial Products. Wrigley S, Hayes M, Thomas R, Chrystal e (Eds), Royal Society of
-
-
Cragg, G.M.1
-
34
-
-
0028221241
-
-
specificity.
-
Taylor PB, Gulp JS, Debouck C, Johnson RK, Palil AD, Woolf DJ: Kinetic and mutational analysis of human-immunodeficiency-virus type-1 reverse transcriptase by inophyllums, a novel class of non-nucleoside inhibitors. J Biol Chem (1994) 269:6325-6331. An investigation of the nature of the inhibition of reverse transcriptase and its specificity.
-
Gulp JS, Debouck C, Johnson RK, Palil AD, Woolf DJ: Kinetic and Mutational Analysis of Human-immunodeficiency-virus Type-1 Reverse Transcriptase by Inophyllums, A Novel Class of Non-nucleoside Inhibitors. J Biol Chem (1994) 269:6325-6331. An Investigation of the Nature of the Inhibition of Reverse Transcriptase and Its
-
-
Taylor, P.B.1
-
35
-
-
33746502690
-
-
(1990).
-
Hoechst AG (Naik RG, Lal B, Rupp RH, Sedlacek HH, Dickneite G, Czech J): New 4H-1-benzopyran-4-one derivatives and pharmaceutical use. EP-00366061-A (1990).
-
(Naik RG, Lal B, Rupp RH, Sedlacek HH, Dickneite G, Czech J): New 4H-1-benzopyran-4-one Derivatives and Pharmaceutical Use. EP-00366061-A
-
-
Hoechst, A.G.1
|