A novel method of preparation of 3-acylimidazo[1,2-a]pyridines

Heterocycles

Volumn 45, Issue 5, 1997, Pages 897-910

  Moutou, Jean Luc ^a   Schmitt, Martine ^a   Collot, Valérie ^a   Bourguignon, Jean Jacques ^a  

^a Laboratoire de Pharmacochimie   (France)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0001358746     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/com-96-7696     Document Type: Article

References (14)

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12. E. Pretsch, T. Clerc, J. Seibl, and W. Simon", "Tables of Spectral Data for Structure Determination of Organic Compounds", 2nd edition, ed. by W. Fresenius, J. F. K. Huber, E. Pungor, G. A. Rechnitz, W. Simon, and Th. S. West, Springer-Verlag, Inc., 1989.
13. The typical compound (2a) has been prepared in a nonambiguous manner by heating 3,5-dibromo-2-aminopyridine with ethyl α-bromo-β-benzoylacetate in DMF at 60°C for 24 h.
14. A. Marsura, C. Luu-Duc, and G. Gellon, Synthesis, 1985, 537, and references cited herein.