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Volumn 1, Issue 2, 1999, Pages 140-150

High-throughput 1H NMR and HPLC characterization of a 96-member substituted methylene malonamic acid library

(7) Hamper, Bruce C a Snyderman, David M a Owen, Thomas J a Scates, Angela M a Owsley, Dennis C a Kesselring, Allen S a Chott, Robert C a

a MONSANTO COMPANY (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0001294727 PISSN: 15204766 EISSN: None Source Type: Journal
DOI: 10.1021/cc9800172 Document Type: Article

Times cited : (44)

References (39)

1
- 0003867851
- Wiley-Liss: New York
- Gordon, E. M.; Kerwin, J. F. Combinatorial Chemistry and Molecular Diversity in Drug Discovery; Wiley-Liss: New York, 1998.
- (1998) Combinatorial Chemistry and Molecular Diversity in Drug Discovery
- Gordon, E.M.¹ Kerwin, J.F.²

2
- 0004290050
- Academic Press: San Diego, CA
- Bunin, B. A. The Combinatorial Index; Academic Press: San Diego, CA, 1998. Nefzi, A.; Ostresh, J. M.; Houghten, R. A. Chem. Rev. 1997, 97, 449-472. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1997, 53, 5643-5678. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1996, 52, 4527-4554.
- (1998) The Combinatorial Index
- Bunin, B.A.¹

3
- 7444256652
- Bunin, B. A. The Combinatorial Index; Academic Press: San Diego, CA, 1998. Nefzi, A.; Ostresh, J. M.; Houghten, R. A. Chem. Rev. 1997, 97, 449-472. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1997, 53, 5643-5678. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1996, 52, 4527-4554.
- (1997) Chem. Rev. , vol.97 , pp. 449-472
- Nefzi, A.¹ Ostresh, J.M.² Houghten, R.A.³

4
- 0031001699
- Bunin, B. A. The Combinatorial Index; Academic Press: San Diego, CA, 1998. Nefzi, A.; Ostresh, J. M.; Houghten, R. A. Chem. Rev. 1997, 97, 449-472. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1997, 53, 5643-5678. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1996, 52, 4527-4554.
- (1997) Tetrahedron , vol.53 , pp. 5643-5678
- Hermkens, P.H.H.¹ Ottenheijm, H.C.J.² Rees, D.C.³

5
- 0029930278
- Bunin, B. A. The Combinatorial Index; Academic Press: San Diego, CA, 1998. Nefzi, A.; Ostresh, J. M.; Houghten, R. A. Chem. Rev. 1997, 97, 449-472. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1997, 53, 5643-5678. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1996, 52, 4527-4554.
- (1996) Tetrahedron , vol.52 , pp. 4527-4554
- Hermkens, P.H.H.¹ Ottenheijm, H.C.J.² Rees, D.C.³

6
- 21544474431
- Kyranos, J. N.; Hogan, J. C., Jr. Anal. Chem. 1998, 70, 389-395. Parlow, J. J.; Flynn, D. L. Tetrahedron 1998, 54, 4013-4031.
- (1998) Anal. Chem. , vol.70 , pp. 389-395
- Kyranos, J.N.¹ Hogan Jr., J.C.²

7
- 0032537038
- Kyranos, J. N.; Hogan, J. C., Jr. Anal. Chem. 1998, 70, 389-395. Parlow, J. J.; Flynn, D. L. Tetrahedron 1998, 54, 4013-4031.
- (1998) Tetrahedron , vol.54 , pp. 4013-4031
- Parlow, J.J.¹ Flynn, D.L.²

8
- 0030202425
- Kibbey, C. E. Mol. Diversity 1996, 1 (4), 247-258. Kohler, M.; Haerdi, W.; Christen, P.; Veuthey, J.-L. Trends Anal. Chem. 1997, 16 (8), 475-484.
- (1996) Mol. Diversity , vol.1 , Issue.4 , pp. 247-258
- Kibbey, C.E.¹

9
- 0031239583
- Kibbey, C. E. Mol. Diversity 1996, 1 (4), 247-258. Kohler, M.; Haerdi, W.; Christen, P.; Veuthey, J.-L. Trends Anal. Chem. 1997, 16 (8), 475-484.
- (1997) Trends Anal. Chem. , vol.16 , Issue.8 , pp. 475-484
- Kohler, M.¹ Haerdi, W.² Christen, P.³ Veuthey, J.-L.⁴

10
- 0001690133
- Hamper, B. C.; Kolodziej, S. A.; Scates, A. M.; Smith, R. G.; Cortez, E. J. Org. Chem. 1998, 63, 708-718.
- (1998) J. Org. Chem. , vol.63 , pp. 708-718
- Hamper, B.C.¹ Kolodziej, S.A.² Scates, A.M.³ Smith, R.G.⁴ Cortez, E.⁵

11
- 0005169347
- Daley, D. J.; Scammell, R. D.; James, D.; Monks, I.; Raso, R.; Ashcroft, A. E.; Hudson, A. J. Am. Biotechnol. Lab. 1997, 15, 24-28.
- (1997) Am. Biotechnol. Lab. , vol.15 , pp. 24-28
- Daley, D.J.¹ Scammell, R.D.² James, D.³ Monks, I.⁴ Raso, R.⁵ Ashcroft, A.E.⁶ Hudson, A.J.⁷

12
- 0032499082
- (a) Hamper, B. C.; Kolodziej, S. A.; Scates, A. M. Tetrahedron Lett. 1998, 39, 2047-2050.
- (1998) Tetrahedron Lett. , vol.39 , pp. 2047-2050
- Hamper, B.C.¹ Kolodziej, S.A.² Scates, A.M.³

13
- 0032401987
- (b) For additional references to Knoevenagel condensations on solid phase, see: Shi, S.; Xiao, X.; Czarnik, A. W. Biotechnol. Bioeng. (Comb. Chem.) 1998, 61, 7-12. MacDonald, A. A.; Dewitt, S. H.; Hogan, E. M.; Ramage, R. Tetrahedron Lett. 1996, 37, 4815-4818. Tietze, L. F.; Steinmetz, A. Angew. Chem., Int. Ed. 1996, 35, 651-652. Tietze, L. F.; Hippe, T.; Steinmetz, A. Synlett 1996, 77, 1043-1044. Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643-4646. Zaragoza, F. Tetrahedron Lett. 1995, 36, 8677-8678.
- (1998) Biotechnol. Bioeng. (Comb. Chem.) , vol.61 , pp. 7-12
- Shi, S.¹ Xiao, X.² Czarnik, A.W.³

14
- 0141856793
- (b) For additional references to Knoevenagel condensations on solid phase, see: Shi, S.; Xiao, X.; Czarnik, A. W. Biotechnol. Bioeng. (Comb. Chem.) 1998, 61, 7-12. MacDonald, A. A.; Dewitt, S. H.; Hogan, E. M.; Ramage, R. Tetrahedron Lett. 1996, 37, 4815-4818. Tietze, L. F.; Steinmetz, A. Angew. Chem., Int. Ed. 1996, 35, 651-652. Tietze, L. F.; Hippe, T.; Steinmetz, A. Synlett 1996, 77, 1043-1044. Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643-4646. Zaragoza, F. Tetrahedron Lett. 1995, 36, 8677-8678.
- (1996) Tetrahedron Lett. , vol.37 , pp. 4815-4818
- MacDonald, A.A.¹ Dewitt, S.H.² Hogan, E.M.³ Ramage, R.⁴

15
- 33748225668
- (b) For additional references to Knoevenagel condensations on solid phase, see: Shi, S.; Xiao, X.; Czarnik, A. W. Biotechnol. Bioeng. (Comb. Chem.) 1998, 61, 7-12. MacDonald, A. A.; Dewitt, S. H.; Hogan, E. M.; Ramage, R. Tetrahedron Lett. 1996, 37, 4815-4818. Tietze, L. F.; Steinmetz, A. Angew. Chem., Int. Ed. 1996, 35, 651-652. Tietze, L. F.; Hippe, T.; Steinmetz, A. Synlett 1996, 77, 1043-1044. Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643-4646. Zaragoza, F. Tetrahedron Lett. 1995, 36, 8677-8678.
- (1996) Angew. Chem., Int. Ed. , vol.35 , pp. 651-652
- Tietze, L.F.¹ Steinmetz, A.²

16
- 1542710212
- (b) For additional references to Knoevenagel condensations on solid phase, see: Shi, S.; Xiao, X.; Czarnik, A. W. Biotechnol. Bioeng. (Comb. Chem.) 1998, 61, 7-12. MacDonald, A. A.; Dewitt, S. H.; Hogan, E. M.; Ramage, R. Tetrahedron Lett. 1996, 37, 4815-4818. Tietze, L. F.; Steinmetz, A. Angew. Chem., Int. Ed. 1996, 35, 651-652. Tietze, L. F.; Hippe, T.; Steinmetz, A. Synlett 1996, 77, 1043-1044. Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643-4646. Zaragoza, F. Tetrahedron Lett. 1995, 36, 8677-8678.
- (1996) Synlett , vol.77 , pp. 1043-1044
- Tietze, L.F.¹ Hippe, T.² Steinmetz, A.³

17
- 0030200397
- (b) For additional references to Knoevenagel condensations on solid phase, see: Shi, S.; Xiao, X.; Czarnik, A. W. Biotechnol. Bioeng. (Comb. Chem.) 1998, 61, 7-12. MacDonald, A. A.; Dewitt, S. H.; Hogan, E. M.; Ramage, R. Tetrahedron Lett. 1996, 37, 4815-4818. Tietze, L. F.; Steinmetz, A. Angew. Chem., Int. Ed. 1996, 35, 651-652. Tietze, L. F.; Hippe, T.; Steinmetz, A. Synlett 1996, 77, 1043-1044. Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643-4646. Zaragoza, F. Tetrahedron Lett. 1995, 36, 8677-8678.
- (1996) Tetrahedron Lett. , vol.37 , pp. 4643-4646
- Gordeev, M.F.¹ Patel, D.V.² Wu, J.³ Gordon, E.M.⁴

18
- 0028789375
- (b) For additional references to Knoevenagel condensations on solid phase, see: Shi, S.; Xiao, X.; Czarnik, A. W. Biotechnol. Bioeng. (Comb. Chem.) 1998, 61, 7-12. MacDonald, A. A.; Dewitt, S. H.; Hogan, E. M.; Ramage, R. Tetrahedron Lett. 1996, 37, 4815-4818. Tietze, L. F.; Steinmetz, A. Angew. Chem., Int. Ed. 1996, 35, 651-652. Tietze, L. F.; Hippe, T.; Steinmetz, A. Synlett 1996, 77, 1043-1044. Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643-4646. Zaragoza, F. Tetrahedron Lett. 1995, 36, 8677-8678.
- (1995) Tetrahedron Lett. , vol.36 , pp. 8677-8678
- Zaragoza, F.¹

19
- 0029952401
- Shahripour, A.; Plummer, M. S.; Lunnery, E.; Para, K. S.; Stankovic, C. J.; Rubin, J. R.; Humblet, C.; Fergus, J. H.; Marks, J. S. Bioorg. Med. Chem. Lett. 1996, 6, 1209-1214.
- (1996) Bioorg. Med. Chem. Lett. , vol.6 , pp. 1209-1214
- Shahripour, A.¹ Plummer, M.S.² Lunnery, E.³ Para, K.S.⁴ Stankovic, C.J.⁵ Rubin, J.R.⁶ Humblet, C.⁷ Fergus, J.H.⁸ Marks, J.S.⁹

20
- 8744296233
- Malonyl derivatives of 6-(α-aminoacylamido)penicillanic acids U.S. Patent 3928324, December 23
- Rosati, R. L. Malonyl derivatives of 6-(α-aminoacylamido)penicillanic acids. U.S. Patent 3928324, December 23, 1975.
- (1975)
- Rosati, R.L.¹

21
- 8744263089
- Blagodyr, M. N. Khim.-Farm. Zh. 1993, 27, 27-29.
- (1993) Khim.-Farm. Zh. , vol.27 , pp. 27-29
- Blagodyr, M.N.¹

22
- 8744257885
- Carbapenem compounds, compositions and methods of treatment PCT Int. Appl. WO 9525108, September 21
- Blizzard, T. A.; Ratcliffe, R. W.; Waddell, S. T.; Szumiloski, S. P.; Wilkening, R. R.; Wildonger, K. J. Carbapenem compounds, compositions and methods of treatment PCT Int. Appl. WO 9525108, September 21, 1995. Dininno, F. P. Bridged biphenyl carbapenem antibacterial compounds. PCT Int. Appl. WO 9503700, February 9, 1995.
- (1995)
- Blizzard, T.A.¹ Ratcliffe, R.W.² Waddell, S.T.³ Szumiloski, S.P.⁴ Wilkening, R.R.⁵ Wildonger, K.J.⁶

23
- 8744313060
- Bridged biphenyl carbapenem antibacterial compounds. PCT Int. Appl. WO 9503700, February 9
- Blizzard, T. A.; Ratcliffe, R. W.; Waddell, S. T.; Szumiloski, S. P.; Wilkening, R. R.; Wildonger, K. J. Carbapenem compounds, compositions and methods of treatment PCT Int. Appl. WO 9525108, September 21, 1995. Dininno, F. P. Bridged biphenyl carbapenem antibacterial compounds. PCT Int. Appl. WO 9503700, February 9, 1995.
- (1995)
- Dininno, F.P.¹

24
- 0001535139
- Rigo, B.; Fasseur, D.; Cauliez, P.; Couturier, D. Tetrahedron Lett. 1989, 30, 3073-3076.
- (1989) Tetrahedron Lett. , vol.30 , pp. 3073-3076
- Rigo, B.¹ Fasseur, D.² Cauliez, P.³ Couturier, D.⁴

25
- 0003423124
- IRL Press at Oxford University Press: Oxford, U.K.
- Atherton, E.; Sheppard, R. C. Solid-Phase Peptide Synthesis; IRL Press at Oxford University Press: Oxford, U.K., 1989; pp 9-21.
- (1989) Solid-Phase Peptide Synthesis , pp. 9-21
- Atherton, E.¹ Sheppard, R.C.²

26
- 0030034999
- (a) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937-940; Rockwell, A.; Melden, M.; Copeland, R. A.; Hardman, K.; Decicco, C. P.; Degrado, W. F. J. Am. Chem. Soc. 1996, 118, 10337-10338.
- (1996) Tetrahedron Lett. , vol.37 , pp. 937-940
- Dressman, B.A.¹ Spangle, L.A.² Kaldor, S.W.³

27
- 0029855561
- (a) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937-940; Rockwell, A.; Melden, M.; Copeland, R. A.; Hardman, K.; Decicco, C. P.; Degrado, W. F. J. Am. Chem. Soc. 1996, 118, 10337-10338.
- (1996) J. Am. Chem. Soc. , vol.118 , pp. 10337-10338
- Rockwell, A.¹ Melden, M.² Copeland, R.A.³ Hardman, K.⁴ Decicco, C.P.⁵ Degrado, W.F.⁶

28
- 0031032613
- (b) Gayo, L. M.; Suto, M. J. Tetrahedron Lett. 1997, 38, 211-214.
- (1997) Tetrahedron Lett. , vol.38 , pp. 211-214
- Gayo, L.M.¹ Suto, M.J.²

29
- 0344016189
- (c) Davies, M.; Bradley, M. Angew. Chem. 1997, 109, 1135-1138.
- (1997) Angew. Chem. , vol.109 , pp. 1135-1138
- Davies, M.¹ Bradley, M.²

30
- 0030478424
- (d) Devraj, R.; Cushman, M. J. Org. Chem. 1996, 61, 9368-9373.
- (1996) J. Org. Chem. , vol.61 , pp. 9368-9373
- Devraj, R.¹ Cushman, M.²

31
- 0030470056
- (e) Rotella, D. P. J. Am. Chem. Soc. 1996, 118, 12246-12247.
- (1996) Am. Chem. Soc. , vol.118 , pp. 12246-12247
- Rotella, D.P.J.¹

32
- 0000248247
- Jones, G. Org. Synth. 1967, 15, 204-599.
- (1967) Org. Synth. , vol.15 , pp. 204-599
- Jones, G.¹

33
- 0030477258
- Balkenhohl, F.; von dem Bussche-Huennefeld, C.; Lansky, A.; Zechel, C. Angew. Chem., Int. Ed. 1996, 35, 2288-2337.
- (1996) Angew. Chem., Int. Ed. , vol.35 , pp. 2288-2337
- Balkenhohl, F.¹ Von Dem Bussche-Huennefeld, C.² Lansky, A.³ Zechel, C.⁴

34
- 0000065164
- Tanaka, M.; Oota, O.; Hiramatsu, H.; Fujiwara, K. Bull. Chem. Soc. Jpn. 1988, 61, 2473-2479.
- (1988) Bull. Chem. Soc. Jpn. , vol.61 , pp. 2473-2479
- Tanaka, M.¹ Oota, O.² Hiramatsu, H.³ Fujiwara, K.⁴

35
- 8744247537
- Solid-phase organic synthesis system with pressure-regulated manifold. U.S. Patent 5792430, August 11
- Hamper, B. C. Solid-phase organic synthesis system with pressure-regulated manifold. U.S. Patent 5792430, August 11, 1998; Chem. Abstr. 1998, 128, 142450.
- (1998)
- Hamper, B.C.¹

36
- 8744268633
- Hamper, B. C. Solid-phase organic synthesis system with pressure-regulated manifold. U.S. Patent 5792430, August 11, 1998; Chem. Abstr. 1998, 128, 142450.
- (1998) Chem. Abstr. , vol.128 , pp. 142450

37
- 0031896915
- Keifer, P. A. Drugs Future 1998, 23, 301. Keifer, P. A. Drug Discovery Today, 1997, 2, 468.
- (1998) Drugs Future , vol.23 , pp. 301
- Keifer, P.A.¹

38
- 0030869479
- Keifer, P. A. Drugs Future 1998, 23, 301. Keifer, P. A. Drug Discovery Today, 1997, 2, 468.
- (1997) Drug Discovery Today , vol.2 , pp. 468
- Keifer, P.A.¹

39
- 58149365344
- Smallcombe, S. H.; Patt, S. L.; Keifer, P. A. J. Magn. Reson. A 1995, 777, 295.
- (1995) J. Magn. Reson. A , vol.777 , pp. 295
- Smallcombe, S.H.¹ Patt, S.L.² Keifer, P.A.³

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