Synthesis of C-5 Benzoyl and Azido Functionalized 2,2′-Dithiobisand 2,2′-Diselenobis(1H-indoles)

Journal of Heterocyclic Chemistry

Volumn 34, Issue 5, 1997, Pages 1399-1405

  Sun, Li ^a   Ronald Rubin, J ^a   Kraker, Alan J ^a   Hollis Showalter, H D ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0001266107     PISSN: 0022152X     EISSN: None     Source Type: Journal    
DOI: 10.1002/jhet.5570340505     Document Type: Article

References (10)

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2. H. D. H. Showalter, A. D. Sercel, B. M. Leja, C. D. Wolfangel, L. A. Ambrose, W. L. Elliott, D. W. Fry, A. J. Kraker, C. T. Howard, G. H. Lu, C. W. Moore, B. J. Roberts, P. W. Vincent, W. A. Denny, and A. M. Thompson, J. Med. Chem., 40, 413 (1997).
3. S. A. Fleming, Tetrahedron, 51, 12479 (1995).
4. N. R. Ayyangar, R. J. Lahoti, K. V. Srinivasan, and T. Daniel, Synthesis, 322 (1991).
5. Made by the procedure described by J. Walker, W. Daisley, and A. H. Beckett, J. Med. Chem., 13, 983 (1970) except that toluene was used in place of benzene in the acylation step.
6. K. Kanakarajan, K. Haider, A. W. Czarnik, Synthesis, 566 (1988).
7. H. Suzuki and K. Takaoka, Chem. Lett., 1733 (1984) and references cited therein.
8. A. H. Beckett, R. W. Diasley, and J. Walker, Tetrahedron, 24, 6093 (1968).
9. M. D. Summers and G. E. Smith, Texas Agricultural Experiment Station Bulletin 1555. Texas A & M University, College Station, Texas, (1987).
10. D. W. Fry, A. J. Kraker, R. C. Connors, W. L. Elliott, J. M. Nelson, H. D. H. Showalter, and W. R. Leopold, Anti-Cancer Drug Design, 9, 331 (1994).