Synthesis and pharmacological activity of metabolites of vasopressin V1 receptor antagonist, OPC-21268

Heterocycles

Volumn 43, Issue 12, 1996, Pages 2627-2642

  Otsubo, Kenji ^a   Matsubara, Jun ^a   Ohtani, Tadaaki ^a   Kawano, Yoshikazu ^a   Kitano, Kazuyoshi ^a   Morita, Seiji ^a   Kondo, Kazumi ^a   Yamamura, Yoshitaka ^a   Uchida, Minoru ^a  

^a OTSUKA PHARMACEUTICAL CO LTD   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0001015534     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/com-96-7584     Document Type: Article

References (6)

1. Y. Yamamura, H. Ogawa, T. Chihara, K. Kondo, T. Onogawa, S. Nakamura, T. Mori, M. Tominaga, and Y. Yabuuchi, Science, 1991, 252, 572.
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3. K. Otsubo, S. Morita, and M. Uchida, Bioorg. & Med. Chem. Lett., 1993, 3, 1633.
4. R. C. Corcoran and J. M. Green, Tetrahedron Lett., 1990, 31, 6827.
5. H. Ogawa, H. Miyamoto, K. Kondo, K. Yamashita, K. Nakaya, M. Tominaga, and Y. Yabuuchi, EP Patent 1990, 382185 (Chem. Abstr., 1991, 114, 81619f)
6. T. Nishi, F. Tabusa, T. Tanaka, T. Shimizu, and K. Nakagawa, Chem. Pharm. Bull., 1985, 33, 1140.