A fischer-indole approach to pyrrolo[2,3-d]pyrimidines

Heterocycles

Volumn 43, Issue 2, 1996, Pages 323-338

  Taylor, Edward C ^a   Hu, Baihua ^a  

^a PRINCETON UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0000876969     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/com-95-7260     Document Type: Article

References (10)

1. R. O. Christopherson and S. D. Lyons, Medicinal Research Reviews, 1990, 10, 505 and references cited therein.
2. E. C. Taylor, D. Kuhnt, C. Shih, S. M. Rinzel, G. B. Grindey, J. Barredo, M. Jannatipour, and R. G. Moran, J. Med. Chem., 1992, 35, 4450.
3. a) D. L. Huges, Org. Prep. Proc. Int., 1993, 25, 609 and references cited therein;
4. b) A. Gangjee, J. Patel, R. L. Kisliuk, and Y. Gaumont, J. Med. Chem., 1992, 35, 3678;
5. C. H. Nguyen, J.-M. Lhoste, F. Lavelle, M.-C. Bissery, and E. Bisagni, J. Med. Chem., 1990, 33, 1519.
6. For an analogous synthesis of methyl 4-(5-hydroxypentyl)benzoate and the derived valeraldehyde, see E. C. Taylor and P. M. Harrington, J. Org. Chem., 1990, 55, 3222.
7. E. C. Taylor and A. J. Cocuzza, J. Org. Chem., 1979, 44, 1125.
8. Z. J. Kaminski, Tetrahedron Lett., 1985, 26, 2901.
9. J. I. DeGraw, P. H. Christie, W. T. Colwell, and F. M. Sirotnak, J. Med. Chem., 1992, 35, 320.
10. E. C. Taylor, W. B. Young, R. Chaudhari, and H. H. Patel, Heterocycles, 1993, 36, 1897.