Functional group transformation: An efficacy-enhancing approach in combinatorial chemistry

Journal of Combinatorial Chemistry

Volumn 1, Issue 4, 1999, Pages 307-316

  Hermkens, Pedro H H ^a   Hamersma, Hans ^a  

^a NV ORGANON   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0000718084     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc990003b     Document Type: Article

References (10)

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3. (b) Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Solid-phase organic reactions. II: a review of the literature Nov 95-Nov 96. Tetrahedron 1997, 53, 5643-5678.
4. (c) Booth, S.; Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Solid-phase organic reactions III: a review of the literature November 1996-December 1997. Tetrahedron 1998, 54, 15385-15444.
5. (d) Brown, R. C. D. Recent developments in solid-phase organic synthesis. Contemp. Org. Synth. 1997, 4, 216-237.
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8. (b) Ostresh, J. M.; Schoner, C. C.; Hamashin, V. T.; Nefzi, A.; Meyer, J.-P.; Houghten, R. A. Solid-phase synthesis of trisubstituted bicyclic guanidines via cyclization of reduced N-acylated dipeptides. J. Org. Chem. 1998, 63, 8622-8623.
9. Pei, Y.; Moos W.H. Post-modifications of peptoid side chains: [3+2] cycloaddition of nitrile oxides with alkenes and alkynes on the solid phase. Tetrahedron Lett. 1994, 35, 5825-5828.
10. Boojamra, C. G.; Burow, K. M.; Thompson, L. A.; Ellman, J. A. Solid-phase synthesis of 1,4-benzodiazepine-2,5-diones. Library preparation and demonstration of synthesis generality. J. Org. Chem. 1997, 62, 1240-1256.