Palladium (0)-catalysed arylations using pyrrole and indole 2-boronic acids

Synlett

Volumn , Issue 9, 1998, Pages 1025-1027

  Johnson, Christopher N ^a   Stemp, Geoffrey ^a   Anand, Neel ^b   Stephen, Susanna C ^b   Gallagher, Timothy ^b  

^a GLAXOSMITHKLINE   (United Kingdom)

^b UNIVERSITY OF BRISTOL   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0000271948     PISSN: 09365214     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-1998-1834     Document Type: Article

References (17)

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2. (b) Boyfield, I.; Coldwell, M. C.; Hadley, M. S.; Healy, M. A. M.; Johnson, C. N.; Nash, D. J.; Riley, G. J.; Scott, E. E.; Smith, S. A.; Stemp, G. Bioorg. Med. Chem. Lett. 1997, 7, 327.
3. (c) Bolton, D.; Boyfield, I.; Coldwell, M. C.; Hadley, M. S.; Johns, A.; Johnson, C. N.; Markwell, R. E.; Nash, D. J.; Riley, G. J.; Scott, E. E.; Smith, S. A.; Stemp, G.; Wadsworth, H. J.; Watts, E. A.; Bioorg. Med. Chem. Lett. 1997, 7, 327.
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13. 3) 1.30 (3 H, t, J = 7 Hz), 1.37 (9 H, s), 3.13 (2 H, q, J = 7 Hz), 3.85 (3 H, s), 6.23 (1 H, m), 6.27 (1 H, m), 6.99 (1 H, d, J = 9 Hz), 7.38 (1 H, m), 7.79 (1 H, d, J = 2 Hz), 7.88 (1 H, dd, J = 9, 2 Hz).
14. 3) 1.37 (18 H, s), 6.17 (4 H, d, J = 3 Hz), 7.37 (2 H, t, J = 3 Hz).
15. 3) 1.24 (18 H, s), 6.65 (2 H, s), 7.25 (2 H, dt, J = 8, 1 Hz), 7.35 (2 H, dt, J = 8, 1 Hz), 7.57 (2 H, d, J = 8 Hz), 8.31 (2H, d, J = 8 Hz).
16. Labadie, S. S.; Teng, E. J. Org. Chem. 1994, 59, 4250.
17. Kondo, Y.; Sakamoto, T.; Takazawa, N.; Yamanaka, H. Heterocycles 1993, 36, 941.