Novel indole-ring construction method for the synthesis of 2-trifluoromethylindoles

Heterocycles

Volumn 42, Issue 2, 1996, Pages 513-516

  Miyashita, Kazuyuki ^a   Tsuchiya, Katsutoshi ^a   Kondoh, Katsunori ^a   Miyabe, Hideto ^a   Imanishi, Takeshi ^a  

^a OSAKA UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0000268625     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/com-95-s82     Document Type: Article

References (20)

1. 1. R. Filler and Y. Kobayashi, 'Biomedicinal Aspects of Fluorine Chemistry,' Kodansha, Tokyo, 1982; R. Filler, in 'Fluorine, the First Hundred Years,' ed. by R. E. Banks, D.W. A. Sharp, and J. C. Tatlaw, Elsevier, New York, 1986, p. 361; N. Ishikawa, 'Biologically Active Organofluorine Compounds,' CMC, Tokyo, 1990.
2. R. Filler and Y. Kobayashi, 'Biomedicinal Aspects of Fluorine Chemistry,' Kodansha, Tokyo, 1982; R. Filler, in 'Fluorine, the First Hundred Years,' ed. by R. E. Banks, D.W. A. Sharp, and J. C. Tatlaw, Elsevier, New York, 1986, p. 361; N. Ishikawa, 'Biologically Active Organofluorine Compounds,' CMC, Tokyo, 1990.
3. R. Filler and Y. Kobayashi, 'Biomedicinal Aspects of Fluorine Chemistry,' Kodansha, Tokyo, 1982; R. Filler, in 'Fluorine, the First Hundred Years,' ed. by R. E. Banks, D.W. A. Sharp, and J. C. Tatlaw, Elsevier, New York, 1986, p. 361; N. Ishikawa, 'Biologically Active Organofluorine Compounds,' CMC, Tokyo, 1990.
4. 2. J. E. Saxton, 'The Alkaloids,' Vol. 8, ed. by R. H. F. Manske, Academic Press, New York, 1965, p. 1; R. A. Glennon, J. Med. Chem., 1986, 30, 1.
5. J. E. Saxton, 'The Alkaloids,' Vol. 8, ed. by R. H. F. Manske, Academic Press, New York, 1965, p. 1; R. A. Glennon, J. Med. Chem., 1986, 30, 1.
6. 3. L. J. Audus, 'Plant Growth Substances,' Leonard Hill, London, 1959; T. C. Moore, 'Biochemistry and Physiology of Plant Hormones,' Springer-Verlag, New York, 1979.
7. L. J. Audus, 'Plant Growth Substances,' Leonard Hill, London, 1959; T. C. Moore, 'Biochemistry and Physiology of Plant Hormones,' Springer-Verlag, New York, 1979.
8. a) M. Yoshida, T. Yoshida, M. Kobayashi, and N. Kamigata, J. Chem. Soc., Perkin Trans, 1, 1989, 909;
9. b) Y. Girard, J. G. Atkinson, P. C. Bélanger, J. J. Fuentes, J. Rokach, C. S. Rooney, D. C. Remy and C. A. Hunt, J. Org. Chem., 1983, 48, 3220; Q.-Y. Chen and Z.-T. Li, J. Chem. Soc., Perkin Trans. 1, 1993, 645.
10. b) Y. Girard, J. G. Atkinson, P. C. Bélanger, J. J. Fuentes, J. Rokach, C. S. Rooney, D. C. Remy and C. A. Hunt, J. Org. Chem., 1983, 48, 3220; Q.-Y. Chen and Z.-T. Li, J. Chem. Soc., Perkin Trans. 1, 1993, 645.
11. Y. Kobayashi, I. Kumadaki, Y. Hirose, and Y. Hanzawa, J. Org. Chem., 1974, 39, 1836.
12. W. Madelung, Ber., 1912, 25, 1128.
13. 3, e) G. Bartoli, M. Bosco, R. Dalpozzo, and P. E. Todesco, J. Chem. Soc., Chem. Commun., 1988, 807; G. Bartoli, G. Palmieri, M. Petrini, M. Bosco, and R. Dalpozzo, Tetrahedron, 1990, 46, 1379.
14. 3, e) G. Bartoli, M. Bosco, R. Dalpozzo, and P. E. Todesco, J. Chem. Soc., Chem. Commun., 1988, 807; G. Bartoli, G. Palmieri, M. Petrini, M. Bosco, and R. Dalpozzo, Tetrahedron, 1990, 46, 1379.
15. 3, e) G. Bartoli, M. Bosco, R. Dalpozzo, and P. E. Todesco, J. Chem. Soc., Chem. Commun., 1988, 807; G. Bartoli, G. Palmieri, M. Petrini, M. Bosco, and R. Dalpozzo, Tetrahedron, 1990, 46, 1379.
16. 3, e) G. Bartoli, M. Bosco, R. Dalpozzo, and P. E. Todesco, J. Chem. Soc., Chem. Commun., 1988, 807; G. Bartoli, G. Palmieri, M. Petrini, M. Bosco, and R. Dalpozzo, Tetrahedron, 1990, 46, 1379.
17. 3, e) G. Bartoli, M. Bosco, R. Dalpozzo, and P. E. Todesco, J. Chem. Soc., Chem. Commun., 1988, 807; G. Bartoli, G. Palmieri, M. Petrini, M. Bosco, and R. Dalpozzo, Tetrahedron, 1990, 46, 1379.
18. 3, e) G. Bartoli, M. Bosco, R. Dalpozzo, and P. E. Todesco, J. Chem. Soc., Chem. Commun., 1988, 807; G. Bartoli, G. Palmieri, M. Petrini, M. Bosco, and R. Dalpozzo, Tetrahedron, 1990, 46, 1379.
19. J. P. Li, K. A. Newlander, and T. O. Yellin, Synthesis, 1988, 73.
20. W. A. Remers, in 'Indoles Part One, The Chemistry of Heterocyclic Compounds,' ed. by Houlihan, Wiley-Interscience, New York, 1972, p. 1.